A Phase I/II Study to Evaluate Safety, Tolerability, Pharmacokinetics and Anti-tumor Activity of WSD0922-FU in Combination With Osimertinib for Patients With Locally Advanced or Metastatic Non- Small Cell Lung Cancer

Status: Recruiting
Location: See location...
Intervention Type: Drug
Study Type: Interventional
Study Phase: Phase 1/Phase 2
SUMMARY

This is a Phase I/II, Open Label Study of WSD0922-FU in Combination with Osimertinib for Patients with Locally Advanced or Metastatic Non-Small Cell Lung Cancer whose disease has progressed with third-generation EGFR-TKI with C797S mutation or is newly diagnosed with CNS metastasis with EGFR Del19 or L858R mutation

Eligibility
Participation Requirements
Sex: All
Minimum Age: 18
Healthy Volunteers: f
View:

• ≥Age 18, gender is not limited;

• Locally advanced or metastatic NSCLC confirmed by pathology;

• Patients who have been genetically tested to carry EGFR sensitive mutations;

• Blood/Tissue samples must be provided for testing;

• Must have a minimum life expectancy of \>= 3 months;

• At least one measurable tumor lesion according to RECIST version 1.1; ● Previous radiotherapy-treated lesions cannot be used as target lesions unless imaging studies show clear progression of the lesions.

• Physical Status (ECOG PS) score was 0-1;

• Have full organ function;

• Eligible patients (male and female) who are fertile must agree to use a reliable contraceptive method ;

• Subjects are required to give informed consent to this study before the experiment and sign a written informed consent voluntarily.

Locations
Other Locations
China
Shanghai East Hospital
RECRUITING
Shanghai
Contact Information
Primary
lily Liu, MD
lily.liu@wayshinebiopharm.com
+8613818880308
Backup
Wei Zhong, PhD
wei.zhong@wayshinebiopharm.com
1-951-547-4692
Time Frame
Start Date: 2025-10-17
Estimated Completion Date: 2029-10-14
Participants
Target number of participants: 48
Treatments
Experimental: Dose escalation (WSD0922-FU and Osimertinib)
Patients receive 80mg Osimertinib PO QD and WSD0922-FU PO QD. Cycles repeat every 21 days in the absence of disease progression or unacceptable toxicity. Patients also undergo CT, MRI, and blood sample collection on study.
Experimental: Dose expansion (WSD0922-FU and Osimertinib)
Patients receive 80mg Osimertinib PO QD and WSD0922-FU PO QD using dosage selected from Dose escalation. Cycles repeat every 21 days in the absence of disease progression or unacceptable toxicity. Patients also undergo CT, MRI, and blood sample collection on study.
Sponsors
Leads: Wayshine Biopharm, Inc.

This content was sourced from clinicaltrials.gov