Estradiol-mediated Inflammation and Central Sensitization in the Pathophysiology of Endometriosis-associated Pelvic Pain

Status: Recruiting
Location: See location...
Intervention Type: Drug
Study Type: Interventional
Study Phase: Phase 3
SUMMARY

The purpose of this study is to better understand how hormone suppression with Relugolix Combination-Therapy (CT) affects pelvic pain, inflammation, and pain sensitivity in women with moderate-to-severe endometriosis associated pelvic pain.

Eligibility
Participation Requirements
Sex: Female
Minimum Age: 21
Maximum Age: 49
Healthy Volunteers: f
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• Premenopausal woman between age 21 and 49 years (inclusive) at the time of consent. Menopause is defined as amenorrhea \>1 year unrelated to hormonal suppression.

• History of endometriosis diagnosed by surgery (visual or biopsy confirmed), ultrasound, or MRI within 5 years of study entry

• History of self-reported moderate to severe pelvic pain for ≥ 6 months' duration at time of screening visit. Moderate-to-severe pelvic pain will be defined as self-report recall of average non-menstrual pelvic pain score over past 6 months as ≥ 4 on a 0-10 numeric rating scale (NRS)

• Willingness to participate in a relugolix CT drug intervention trial

• No use of adjunctive pain medications or on stable chronic daily use of adjunctive pain medications (excluding opioids);

• Has not used an injectable hormone therapy in the past 6 months (e.g. DepoProvera®, DepoLupron®).

• Willingness to 30-60 day washout interval of oral, vaginal, transdermal, intrauterine hormonal therapies prior to study initiation if applicable

• Willingness to use 2 forms of non-hormonal contraception during the entire duration of the study period or has had a history of a bilateral tubal occlusion procedure at least 3 months prior to screening (tubal ligation or hysteroscopic occlusion method)

• Willing to undergo quantitative sensory testing (QST), fMRI and other study procedures

• Ability to read and speak English to allow for written informed consent, phenotyping, and patient-reported outcomes measures

• Meet criteria to participate in QST and fMRI. These include:

• Normal visual acuity or correctable (with corrective lenses- glasses or contacts) to at least 20/40 for reading instructions in the MRI and visual sensitivity testing

• No contraindications to MRI (e.g., metal implants, claustrophobia)

• Willingness to refrain from pain medications such as NSAIDs, acetaminophen, and opioids for 12 hours prior to neuroimaging and QST

• Willingness to refrain from alcohol and nicotine on day of QST and neuroimaging (alcohol and nicotine consumption is allowed after testing is completed)

• Willingness to refrain from physical activity or exercise that would cause muscle and/or joint soreness for 48 hours prior to testing (routine exercise or activity that does not lead to soreness is acceptable)

• Able to lie still on their back for 1 hour during MRI

Locations
United States
Michigan
University of Michigan
RECRUITING
Ann Arbor
Contact Information
Primary
Kathy Scott
jrsj@med.umich.edu
734-998-7022
Time Frame
Start Date: 2025-11
Estimated Completion Date: 2028-09
Participants
Target number of participants: 130
Treatments
Experimental: Relugolix CT
All participants will have the same intervention, but approximately half of those enrolled will have widespread pain and half will not.~Approximately 65 participants with widespread pain will receive relugolix CT (relugolix 40mg, estradiol 1 mg, norethindrone acetate 0.5 mg once daily) daily for 24 weeks, and 65 participants without widespread pain will receive relugolix CT for 24 weeks.
Related Therapeutic Areas
Sponsors
Leads: University of Michigan
Collaborators: Eunice Kennedy Shriver National Institute of Child Health and Human Development (NICHD)

This content was sourced from clinicaltrials.gov

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