An Open-label Study to Assess the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of GT-02287 in Participants With Parkinson's Disease With or Without a Pathogenic GBA1 Mutation

Status: Recruiting
Location: See all (7) locations...
Intervention Type: Drug
Study Type: Interventional
Study Phase: Phase 1
SUMMARY

The main goal of this clinical trial is to learn about the safety and tolerability of GT-02287. The questions it aims to answer are: * What medical problems do participants have when taking GT-02287? * How is GT-02287 absorbed, distributed, and removed from the body of participants over time (pharmacokinetics)? * Are there any biological effects of GT-02287 in blood and in cerebrospinal fluid that could be beneficial for people with Parkinson's disease? Participants will: * visit the clinic to assess if they qualify for the study (30-day Screening Period) * if eligible, receive GT-02287 once a day every day for 90 days (90-day Open Label Treatment period) * visit the clinic the first day of treatment, after the first 2 weeks of treatment, and every month during the 90-day Treatment Period. * visit the clinic to assess how they are doing 14 days after the end of GT-02287 treatment (14-day Follow-Up Period).

Eligibility
Participation Requirements
Sex: All
Minimum Age: 30
Maximum Age: 85
Healthy Volunteers: f
View:

• Able and willing to provide written informed consent and be willing to comply with the requirements and restrictions of the study

• Any sex, ≥30 and ≤85 years of age

• Diagnosis of PD based on MDS criteria

• Within 7 years of PD diagnosis

• Body mass index of ≥18 and ≤40 kg/m2, and a body weight ≥45 kg and ≤120 kg

• Willing to provide a blood sample for PD-related genetic testing

• Hoehn \& Yahr 1-3, inclusive

• No severe motor fluctuations or disabling dyskinesias based on the investigator's clinical assessment

• Naïve to pharmacological treatment for PD or on stable PD medication for ≥3 months prior to Screening, including ≥4 weeks at the same dose(s) immediately before Screening

• Not pregnant or breastfeeding

• If participant is either of childbearing potential or produces potentially viable sperm, participant must agree to use 2 forms of contraception (barrier method and a second highly effective form of birth control/contraception, as defined in the protocol) if engaging in potentially reproductive intercourse (with a partner who produces potentially viable sperm or is of childbearing potential, respectively)

• Agreeing to not participate in another investigational study while taking part in this study

• For participants with known GBA1 mutations, presence of a GBA1 mutation that has been associated with an increased risk of PD

Locations
Other Locations
Australia
CMAX
RECRUITING
Adelaide
St Vincent's Hospital Sydney
RECRUITING
Darlinghurst
Southern Neurology
RECRUITING
Kogarah
Alfred Health
RECRUITING
Melbourne
Royal Melbourne Hospital
RECRUITING
Parkville
Westmead Hospital
RECRUITING
Westmead
Princess Alexandra Hospital
RECRUITING
Woolloongabba
Contact Information
Primary
Gain Therapeutics Clinical Operations
info@gaintherapeutics.com
+41919211131
Time Frame
Start Date: 2025-02-21
Estimated Completion Date: 2025-11-30
Participants
Target number of participants: 20
Treatments
Experimental: single-arm. All participants receive the active molecule (once daily GT-02287 administration)
Related Therapeutic Areas
Sponsors
Leads: Gain Therapeutics, Inc.

This content was sourced from clinicaltrials.gov