Adrien Delpal

Marseille, France

Last Updated: 09/26/2026

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Found 14 publications

Crystallographic characterisation and development of bi-substrate inhibitors of coronavirus nsp14 methyltransferase.

Crystallographic characterisation and development of bi-substrate inhibitors of coronavirus nsp14 methyltransferase.

Journal: RSC medicinal chemistry

Published: October 08, 2025

Synthesis and in vitro inhibitory activity of N-arylsulfonamide adenosine analogues designed to target SARS-CoV-2 nsp14 N7-methyltransferase.

Synthesis and in vitro inhibitory activity of N-arylsulfonamide adenosine analogues designed to target SARS-CoV-2 nsp14 N7-methyltransferase.

Journal: Bioorganic chemistry

Published: July 22, 2025

N-Arylsulfonamide-based adenosine analogues to target RNA cap N7-methyltransferase nsp14 of SARS-CoV-2.

N-Arylsulfonamide-based adenosine analogues to target RNA cap N7-methyltransferase nsp14 of SARS-CoV-2.

Journal: RSC medicinal chemistry

Published: December 22, 2023

5'-cap RNA/SAM mimetic conjugates as bisubstrate inhibitors of viral RNA cap 2'-O-methyltransferases.

5'-cap RNA/SAM mimetic conjugates as bisubstrate inhibitors of viral RNA cap 2'-O-methyltransferases.

Journal: Bioorganic chemistry

Published: October 23, 2023

Structure-guided optimization of adenosine mimetics as selective and potent inhibitors of coronavirus nsp14 N7-methyltransferases.

Structure-guided optimization of adenosine mimetics as selective and potent inhibitors of coronavirus nsp14 N7-methyltransferases.

Journal: European journal of medicinal chemistry

Published: February 16, 2023

Facile access to 4'-(N-acylsulfonamide) modified nucleosides and evaluation of their inhibitory activity against SARS-CoV-2 RNA cap N7-guanine-methyltransferase nsp14.

Facile access to 4'-(N-acylsulfonamide) modified nucleosides and evaluation of their inhibitory activity against SARS-CoV-2 RNA cap N7-guanine-methyltransferase nsp14.

Journal: Organic & biomolecular chemistry

Published: September 26, 2022

A Versatile Class of 1,4,4-Trisubstituted Piperidines Block Coronavirus Replication In Vitro.

A Versatile Class of 1,4,4-Trisubstituted Piperidines Block Coronavirus Replication In Vitro.

Journal: Pharmaceuticals (Basel, Switzerland)

Published: July 26, 2022

Erratum for Essalmani et al., "Distinctive Roles of Furin and TMPRSS2 in SARS-CoV-2 Infectivity".

Erratum for Essalmani et al., "Distinctive Roles of Furin and TMPRSS2 in SARS-CoV-2 Infectivity".

Journal: Journal of virology

Published: June 06, 2022

Design and synthesis of naturally-inspired SARS-CoV-2 inhibitors.

Design and synthesis of naturally-inspired SARS-CoV-2 inhibitors.

Journal: RSC medicinal chemistry

Published: May 18, 2022

Potent Inhibition of SARS-CoV-2 nsp14 N7-Methyltransferase by Sulfonamide-Based Bisubstrate Analogues.

Potent Inhibition of SARS-CoV-2 nsp14 N7-Methyltransferase by Sulfonamide-Based Bisubstrate Analogues.

Journal: Journal of medicinal chemistry

Published: April 19, 2022

Distinctive Roles of Furin and TMPRSS2 in SARS-CoV-2 Infectivity.

Distinctive Roles of Furin and TMPRSS2 in SARS-CoV-2 Infectivity.

Journal: Journal of virology

Published: March 28, 2022

Synthesis, Structure-Activity Relationships, and Antiviral Profiling of 1-Heteroaryl-2-Alkoxyphenyl Analogs as Inhibitors of SARS-CoV-2 Replication.

Synthesis, Structure-Activity Relationships, and Antiviral Profiling of 1-Heteroaryl-2-Alkoxyphenyl Analogs as Inhibitors of SARS-CoV-2 Replication.

Journal: Molecules (Basel, Switzerland)

Published: December 20, 2021

Showing 1-12 of 14

Last Updated: 09/26/2026