Akira Otaka

Tokushima, 7708505, Japan

Last Updated: 09/26/2026

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Found 76 publications

2-Mercaptophenylboronic acid: a superior alternative to 2-mercaptoethanol for thioester hydrolysis.

2-Mercaptophenylboronic acid: a superior alternative to 2-mercaptoethanol for thioester hydrolysis.

Journal: Organic & biomolecular chemistry

Published: April 27, 2026

A one-step, resin-compatible Cys-Trp cross-linking system opens a new avenue for stapled peptide therapeutics.

A one-step, resin-compatible Cys-Trp cross-linking system opens a new avenue for stapled peptide therapeutics.

Journal: Bioorganic & medicinal chemistry

Published: February 05, 2026

Late-Stage Intermolecular O-Peptidylation Protocol Enabled by Sequential Acyl Transfer on Thiol-Incorporated Threonine Followed by Desulfurization.

Late-Stage Intermolecular O-Peptidylation Protocol Enabled by Sequential Acyl Transfer on Thiol-Incorporated Threonine Followed by Desulfurization.

Journal: Chemistry (Weinheim an der Bergstrasse, Germany)

Published: March 18, 2025

Late-Stage Formation of a Sactionine Linkage Enabled by Lossen Rearrangement of Glycyl Hydroxamic Acid.

Late-Stage Formation of a Sactionine Linkage Enabled by Lossen Rearrangement of Glycyl Hydroxamic Acid.

Journal: Organic letters

Published: June 07, 2024

Synthesis of N-Glyoxylyl Peptides Enabled by a Lossen Rearrangement-Induced Intramolecular Redox Reaction of N-Terminal Glycyl Hydroxamic Acid.

Synthesis of N-Glyoxylyl Peptides Enabled by a Lossen Rearrangement-Induced Intramolecular Redox Reaction of N-Terminal Glycyl Hydroxamic Acid.

Journal: Organic letters

Published: May 13, 2024

Cysteinylprolyl ester-mediated drug release from a lipid-drug conjugate.

Cysteinylprolyl ester-mediated drug release from a lipid-drug conjugate.

Journal: Bioorganic & medicinal chemistry letters

Published: April 30, 2024

Advanced Insulin Synthesis by One-pot/Stepwise Disulfide Bond Formation Enabled by S-Protected Cysteine Sulfoxide.

Advanced Insulin Synthesis by One-pot/Stepwise Disulfide Bond Formation Enabled by S-Protected Cysteine Sulfoxide.

Journal: Chemistry (Weinheim an der Bergstrasse, Germany)

Published: March 11, 2024

Identification of Low-Density Lipoprotein Receptor-Related Protein 1 as a CXCL14 Receptor Using Chemically Synthesized Tetrafunctional Probes.

Identification of Low-Density Lipoprotein Receptor-Related Protein 1 as a CXCL14 Receptor Using Chemically Synthesized Tetrafunctional Probes.

Journal: ACS chemical biology

Published: January 30, 2024

Effects of tryptophan-selective lipidated glucagon-like peptide 1 (GLP-1) peptides on the GLP-1 receptor.

Effects of tryptophan-selective lipidated glucagon-like peptide 1 (GLP-1) peptides on the GLP-1 receptor.

Journal: The Journal of endocrinology

Published: January 24, 2024

Enhanced tumor specific drug release by hypoxia sensitive dual-prodrugs based on 2-nitroimidazole.

Enhanced tumor specific drug release by hypoxia sensitive dual-prodrugs based on 2-nitroimidazole.

Journal: Bioorganic & medicinal chemistry letters

Published: July 04, 2023

CA9 and PRELID2; hypoxia-responsive potential therapeutic targets for pancreatic ductal adenocarcinoma as per bioinformatics analyses.

CA9 and PRELID2; hypoxia-responsive potential therapeutic targets for pancreatic ductal adenocarcinoma as per bioinformatics analyses.

Journal: Journal of pharmacological sciences

Published: May 28, 2023

Residue-Selective C-H Sulfenylation Enabled by Acid-Activated S-Acetamidomethyl Cysteine Sulfoxide with Application to One-Pot Stapling and Lipidation Sequence.

Residue-Selective C-H Sulfenylation Enabled by Acid-Activated S-Acetamidomethyl Cysteine Sulfoxide with Application to One-Pot Stapling and Lipidation Sequence.

Journal: Chemistry (Weinheim an der Bergstrasse, Germany)

Published: March 12, 2023

Showing 1-12 of 76

Last Updated: 09/26/2026