Andrew P. Montgomery
Sydney, NSW 2006, Australia
Last Updated: 09/26/2026
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Found 25 publications
Erratum to 'The discovery of a potent and selective pyrazolo-[2,3-e]-[1,2,4]-triazine cannabinoid type 2 receptor agonist' [Eur. J. Med. Chem. 210 (2021) 113087].
Journal: European journal of medicinal chemistry
Published: April 09, 2026
The adamantane scaffold: Beyond a lipophilic moiety.
Journal: European journal of medicinal chemistry
Published: February 11, 2025
Histone methyltransferase PRDM9 promotes survival of drug-tolerant persister cells in glioblastoma.
Journal: Nature communications
Published: October 17, 2024
PK 11195 derivatives: exploring the influence of amide and heterocyclic substitution on A147T TSPO discrimination.
Journal: RSC medicinal chemistry
Published: October 14, 2024
Enhancing CNS mitophagy: drug development and disease-relevant models.
Journal: Trends in pharmacological sciences
Published: August 02, 2024
Structure-based drug design for TSPO: Challenges and opportunities.
Journal: Biochimie
Published: February 19, 2024
Fragment-based drug discovery for disorders of the central nervous system: designing better drugs piece by piece.
Journal: Frontiers in chemistry
Published: January 31, 2024
Synthesis of α-Hydroxy-1,2,3-Triazole-linked Sialyltransferase Inhibitors and Evaluation of Selectivity Towards ST3GAL1, ST6GAL1 and ST8SIA2.
Journal: ChemMedChem
Published: January 30, 2024
Efficacy of DYRK1A inhibitors in novel models of Down syndrome acute lymphoblastic leukemia.
Journal: Haematologica
Published: September 13, 2023
Synthesis and Preclinical Evaluation of Fluorinated 5-Azaindoles as CB2 PET Radioligands.
Journal: ACS chemical neuroscience
Published: July 27, 2023
Late-stage Functionalization for Improving Drug-like Molecular Properties.
Journal: Chemical reviews
Published: June 07, 2023
An update on late-stage functionalization in today's drug discovery.
Journal: Expert opinion on drug discovery
Published: April 28, 2023
Last Updated: 09/26/2026