Angelique Mularoni

Lyon, France

Last Updated: 09/26/2026

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Found 13 publications

Targeting Human Protein Kinase CK2 by a Library of Indeno[1,2-b]Indoles: Contribution of Thermal Shift Assay to Pre-Screening and Co-Crystallization to Post-Screening.

Targeting Human Protein Kinase CK2 by a Library of Indeno[1,2-b]Indoles: Contribution of Thermal Shift Assay to Pre-Screening and Co-Crystallization to Post-Screening.

Journal: Archiv der Pharmazie
Published: March 04, 2026

Discovery of KDX1381, a Bivalent CK2α Inhibitor for the Treatment of Solid Tumors as a Single Agent or in Combination.

Discovery of KDX1381, a Bivalent CK2α Inhibitor for the Treatment of Solid Tumors as a Single Agent or in Combination.

Journal: Journal of medicinal chemistry
Published: June 10, 2025

Picomolar bivalent inhibitors of protein kinase CK2 active against β-coronavirus replication.

Picomolar bivalent inhibitors of protein kinase CK2 active against β-coronavirus replication.

Journal: European journal of medicinal chemistry
Published: April 16, 2025

Exploring the biological potential of the brominated indenoindole MC11 and its interaction with protein kinase CK2.

Exploring the biological potential of the brominated indenoindole MC11 and its interaction with protein kinase CK2.

Journal: Biological chemistry
Published: December 15, 2024

Binding-Site Switch for Protein Kinase CK2 Inhibitors.

Binding-Site Switch for Protein Kinase CK2 Inhibitors.

Journal: ChemMedChem
Published: October 30, 2024

Design, synthesis, and structure-activity relationship studies of 6H-benzo[b]indeno[1,2-d]thiophen-6-one derivatives as DYRK1A/CLK1/CLK4/haspin inhibitors.

Design, synthesis, and structure-activity relationship studies of 6H-benzo[b]indeno[1,2-d]thiophen-6-one derivatives as DYRK1A/CLK1/CLK4/haspin inhibitors.

Journal: RSC medicinal chemistry
Published: July 13, 2024

Cancer selective cell death induction by a bivalent CK2 inhibitor targeting the ATP site and the allosteric αD pocket.

Cancer selective cell death induction by a bivalent CK2 inhibitor targeting the ATP site and the allosteric αD pocket.

Journal: iScience
Published: April 19, 2023

Combining nano-differential scanning fluorimetry and microscale thermophoresis to investigate VDAC1 interaction with small molecules.

Combining nano-differential scanning fluorimetry and microscale thermophoresis to investigate VDAC1 interaction with small molecules.

Journal: Journal of enzyme inhibition and medicinal chemistry
Published: January 18, 2023

Tetanus Toxin Fragment C: Structure, Drug Discovery Research and Production.

Tetanus Toxin Fragment C: Structure, Drug Discovery Research and Production.

Journal: Pharmaceuticals (Basel, Switzerland)
Published: May 20, 2022

Synthesis, Optimization, Antifungal Activity, Selectivity, and CYP51 Binding of New 2-Aryl-3-azolyl-1-indolyl-propan-2-ols.

Synthesis, Optimization, Antifungal Activity, Selectivity, and CYP51 Binding of New 2-Aryl-3-azolyl-1-indolyl-propan-2-ols.

Journal: Pharmaceuticals (Basel, Switzerland)
Published: July 15, 2020

N,N'-disubstituted cinnamamide derivatives potentiate ciprofloxacin activity against overexpressing NorA efflux pump Staphylococcus aureus 1199B strains.

N,N'-disubstituted cinnamamide derivatives potentiate ciprofloxacin activity against overexpressing NorA efflux pump Staphylococcus aureus 1199B strains.

Journal: European journal of medicinal chemistry
Published: December 05, 2017

Screening of indeno[1,2-b]indoloquinones by MALDI-MS: a new set of potential CDC25 phosphatase inhibitors brought to light.

Screening of indeno[1,2-b]indoloquinones by MALDI-MS: a new set of potential CDC25 phosphatase inhibitors brought to light.

Journal: Journal of enzyme inhibition and medicinal chemistry
Published: July 01, 2016
Showing 1-12 of 13

Last Updated: 09/26/2026