Anthony Bouillon
Paris, France
Last Updated: 09/26/2026
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Found 10 publications
Towards Improved Peptidic α-Ketoamide Inhibitors of the Plasmodial Subtilisin-Like SUB1: Exploration of N-Terminal Extensions and Cyclic Constraints.
Journal: ChemMedChem
Published: November 15, 2024
Prodomain-driven enzyme dimerization: a pH-dependent autoinhibition mechanism that controls Plasmodium Sub1 activity before merozoite egress.
Journal: mBio
Published: February 22, 2024
Insights from structure-activity relationships and the binding mode of peptidic α-ketoamide inhibitors of the malaria drug target subtilisin-like SUB1.
Journal: European journal of medicinal chemistry
Published: December 11, 2023
3D structures of the Plasmodium vivax subtilisin-like drug target SUB1 reveal conformational changes to accommodate a substrate-derived α-ketoamide inhibitor.
Journal: Acta crystallographica. Section D, Structural biology
Published: March 13, 2023
Prevalence and characterization of piperaquine, mefloquine and artemisinin derivatives triple-resistant Plasmodium falciparum in Cambodia.
Journal: The Journal of antimicrobial chemotherapy
Published: July 13, 2022
A surrogate marker of piperaquine-resistant Plasmodium falciparum malaria: a phenotype-genotype association study.
Journal: The Lancet. Infectious diseases
Published: August 12, 2016
Computational design of protein-based inhibitors of Plasmodium vivax subtilisin-like 1 protease.
Journal: PloS one
Published: April 18, 2014
A novel Plasmodium-specific prodomain fold regulates the malaria drug target SUB1 subtilase.
Journal: Nature communications
Published: March 06, 2014
In Silico screening on the three-dimensional model of the Plasmodium vivax SUB1 protease leads to the validation of a novel anti-parasite compound.
Journal: The Journal of biological chemistry
Published: May 09, 2013
Screening and evaluation of inhibitors of Plasmodium falciparum merozoite egress and invasion using cytometry.
Journal: Methods in molecular biology (Clifton, N.J.)
Published: September 20, 2012
Showing 1-10 of 10
Last Updated: 09/26/2026