Antimo Gioiello
Perugia, 06123, Italy
Last Updated: 09/26/2026
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Found 76 publications
Lighting Up Gut Dysbiosis: Red-Shifted Whole-Cell Bioluminescence Enables Functional Sensing of Bile Salt Hydrolase Activity in Human Feces.
Journal: ACS sensors
Published: June 12, 2026
Advanced Synthetic Methods in Modern Medicinal Chemistry.
Journal: Journal of medicinal chemistry
Published: May 28, 2026
Development of Biphenyl-Substituted Uracil-Based Hydroxamic Acids (UBHAs) as Potent HDAC Inhibitors with Pro-Apoptotic Activity in Leukemia and Prostate Cancer Cells.
Journal: Journal of medicinal chemistry
Published: April 30, 2026
Development of Biphenyl-Substituted Uracil-Based Hydroxamic Acids (UBHAs) as Potent HDAC Inhibitors with Pro-Apoptotic Activity in Leukemia and Prostate Cancer Cells.
Journal: Journal of medicinal chemistry
Published: April 30, 2026
Garcinoic acid: A vitamin E metabolite-mimetic scaffold linking nuclear receptor pharmacology to inflammatory signaling and biomimetic drug discovery.
Journal: Pharmacology & therapeutics
Published: April 18, 2026
Lipid nanoparticles for Ursodeoxycholic Acid Delivery: A Strategy for Topical Applications.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences
Published: April 08, 2026
The rare bile acid isoallolithocholic acid (IALCA) is an EphA2 antagonist sparing FXR and TGR5 receptors.
Journal: Biochemical pharmacology
Published: December 18, 2025
Novel tyrosinol-based chiral stationary phase for the separation of tetracyclic quinolines active as PXR agonists: Investigating the enantiorecognition mechanism through molecular dynamics.
Journal: Analytica chimica acta
Published: October 28, 2025
Structure-Based Discovery of Obeticholic Acid Derivatives as Novel Farnesoid X Receptor Partial Agonists with Improved Selectivity and Reduced Off-Target Effects.
Journal: ChemMedChem
Published: October 24, 2025
Novel Sulfonium Reagents for the Modular Synthesis of Spiro[2.3]Hexanes and Heteroatom-Containing Analogues: Synthesis, Application, and Evaluation as Bioisosteres.
Journal: Angewandte Chemie (International ed. in English)
Published: October 02, 2025
Discovery and development of steroidal enzyme inhibitors as anti-cancer drugs: state-of-the-art and future perspectives.
Journal: Journal of enzyme inhibition and medicinal chemistry
Published: April 02, 2025
Garcinoic acid enhances inflammation resolution against colitis by activating Nrf2 dependent efferocytosis.
Journal: Free radical biology & medicine
Published: January 31, 2025
Last Updated: 09/26/2026