Antonio J. Vargas-Moreno

Sevilla, AN 41012, Spain

Last Updated: 09/26/2026

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Found 26 publications

Glutathione-Responsive Fragmentation of Heteronorbornadiene-Based Thiovinyl Sulfones in Glioma Cells.

Glutathione-Responsive Fragmentation of Heteronorbornadiene-Based Thiovinyl Sulfones in Glioma Cells.

Journal: Bioconjugate chemistry

Published: April 28, 2026

[2.2.1]Heterobicyclic Bromovinyl Sulfones for Thiol-Triggered Strategies in Linker Chemistry: Aza- vs Oxa-Norbornadienic Systems.

[2.2.1]Heterobicyclic Bromovinyl Sulfones for Thiol-Triggered Strategies in Linker Chemistry: Aza- vs Oxa-Norbornadienic Systems.

Journal: Bioconjugate chemistry

Published: August 22, 2025

Experimental and Theoretical Analysis of the Thiol-Promoted Fragmentation of 2-Halo-3-tosyl-oxanorbornadienes.

Experimental and Theoretical Analysis of the Thiol-Promoted Fragmentation of 2-Halo-3-tosyl-oxanorbornadienes.

Journal: Organic letters

Published: October 10, 2023

Synthesis and structure-activity relationship of new nicotinamide phosphoribosyltransferase inhibitors with antitumor activity on solid and haematological cancer.

Synthesis and structure-activity relationship of new nicotinamide phosphoribosyltransferase inhibitors with antitumor activity on solid and haematological cancer.

Journal: European journal of medicinal chemistry

Published: January 10, 2023

Identification of new FK866 analogues with potent anticancer activity against pancreatic cancer.

Identification of new FK866 analogues with potent anticancer activity against pancreatic cancer.

Journal: European journal of medicinal chemistry

Published: February 02, 2022

Carbohydrate-derived bicyclic selenazolines as new dual inhibitors (cholinesterases/OGA) against Alzheimer's disease.

Carbohydrate-derived bicyclic selenazolines as new dual inhibitors (cholinesterases/OGA) against Alzheimer's disease.

Journal: Bioorganic chemistry

Published: December 19, 2021

Discovery of human hexosaminidase inhibitors by in situ screening of a library of mono- and divalent pyrrolidine iminosugars.

Discovery of human hexosaminidase inhibitors by in situ screening of a library of mono- and divalent pyrrolidine iminosugars.

Journal: Bioorganic chemistry

Published: December 09, 2021

Synthesis of multimeric pyrrolidine iminosugar inhibitors of human β-glucocerebrosidase and α-galactosidase A: First example of a multivalent enzyme activity enhancer for Fabry disease.

Synthesis of multimeric pyrrolidine iminosugar inhibitors of human β-glucocerebrosidase and α-galactosidase A: First example of a multivalent enzyme activity enhancer for Fabry disease.

Journal: European journal of medicinal chemistry

Published: November 21, 2019

Stable Pyrrole-Linked Bioconjugates through Tetrazine-Triggered Azanorbornadiene Fragmentation.

Stable Pyrrole-Linked Bioconjugates through Tetrazine-Triggered Azanorbornadiene Fragmentation.

Journal: Angewandte Chemie (International ed. in English)

Published: November 13, 2019

Structural basis of the inhibition of GH1 β-glucosidases by multivalent pyrrolidine iminosugars.

Structural basis of the inhibition of GH1 β-glucosidases by multivalent pyrrolidine iminosugars.

Journal: Bioorganic chemistry

Published: May 02, 2019

Dual targeting of PTP1B and glucosidases with new bifunctional iminosugar inhibitors to address type 2 diabetes.

Dual targeting of PTP1B and glucosidases with new bifunctional iminosugar inhibitors to address type 2 diabetes.

Journal: Bioorganic chemistry

Published: January 15, 2019

Azabicyclic vinyl sulfones for residue-specific dual protein labelling.

Azabicyclic vinyl sulfones for residue-specific dual protein labelling.

Journal: Chemical science

Published: January 09, 2019

Showing 1-12 of 26

Last Updated: 09/26/2026