Arthur Christopoulos

Parkville, VIC 3052, Australia

Last Updated: 09/26/2026

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Found 258 publications

The Design, Synthesis and Pharmacological Characterization of Potent Xanomeline-Based M1 and M4 mAChR Bitopic Ligands.

The Design, Synthesis and Pharmacological Characterization of Potent Xanomeline-Based M1 and M4 mAChR Bitopic Ligands.

Journal: Journal of medicinal chemistry
Published: July 27, 2026

Low Agonism and Balanced Pathway Modulation Distinguish an M1 Muscarinic Receptor Positive Allosteric Modulator Lacking Cholinergic Adverse Effects.

Low Agonism and Balanced Pathway Modulation Distinguish an M1 Muscarinic Receptor Positive Allosteric Modulator Lacking Cholinergic Adverse Effects.

Journal: ACS chemical neuroscience
Published: June 30, 2026

The Concise Guide to PHARMACOLOGY 2025/26: G protein-coupled receptors.

The Concise Guide to PHARMACOLOGY 2025/26: G protein-coupled receptors.

Journal: British journal of pharmacology
Published: December 29, 2025

Structure-guided allosteric modulation of the delta opioid receptor.

Structure-guided allosteric modulation of the delta opioid receptor.

Journal: bioRxiv : the preprint server for biology
Published: November 24, 2025

Dissociation kinetics of G proteins from G protein-coupled receptors and effects of allosteric modulation.

Dissociation kinetics of G proteins from G protein-coupled receptors and effects of allosteric modulation.

Journal: Proceedings of the National Academy of Sciences of the United States of America
Published: November 13, 2025

Structure-Activity Relationships of Highly Potent and Selective A2B Adenosine Receptor Agonists.

Structure-Activity Relationships of Highly Potent and Selective A2B Adenosine Receptor Agonists.

Journal: Journal of medicinal chemistry
Published: October 23, 2025

A Structure-Activity Relationship Study of Novel Positive Allosteric Modulators for the δ-Opioid Receptor.

A Structure-Activity Relationship Study of Novel Positive Allosteric Modulators for the δ-Opioid Receptor.

Journal: ACS chemical neuroscience
Published: July 18, 2025

Structure-based discovery of positive allosteric modulators of the A1 adenosine receptor.

Structure-based discovery of positive allosteric modulators of the A1 adenosine receptor.

Journal: Proceedings of the National Academy of Sciences of the United States of America
Published: July 07, 2025

Reimagining pharmacology education.

Reimagining pharmacology education.

Journal: Pharmacological reviews
Published: June 11, 2025

The Prosperity and Adversity of M4 Muscarinic Acetylcholine Receptor Activators in the Treatment of Neuropsychiatric Disorders.

The Prosperity and Adversity of M4 Muscarinic Acetylcholine Receptor Activators in the Treatment of Neuropsychiatric Disorders.

Journal: Journal of medicinal chemistry
Published: April 16, 2025

Cryo-EM reveals a new allosteric binding site at the M5 mAChR.

Cryo-EM reveals a new allosteric binding site at the M5 mAChR.

Journal: bioRxiv : the preprint server for biology
Published: February 20, 2025

Cryo-EM reveals an extrahelical allosteric binding site at the M5 mAChR.

Cryo-EM reveals an extrahelical allosteric binding site at the M5 mAChR.

Journal: Nature communications
Published: February 05, 2025
Showing 1-12 of 258

Last Updated: 09/26/2026