Arturo Galvani
Nerviano, Italy
Last Updated: 09/26/2026
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Found 30 publications
Stereoselective synthesis of 3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-one derivatives as PIM kinase inhibitors inspired from marine alkaloids.
Journal: Chirality
Published: May 14, 2022
Identification of unprecedented ATP-competitive choline kinase inhibitors.
Journal: Bioorganic & medicinal chemistry letters
Published: April 27, 2021
Correction to Discovery of Entrectinib: A New 3-Aminoindazole as a Potent Anaplastic Lymphoma Kinase (ALK), c-ros Oncogene 1 Kinase (ROS1), and Pan-Tropomyosin Receptor Kinases (Pan-TRKs) inhibitor.
Journal: Journal of medicinal chemistry
Published: August 20, 2019
Discovery of Stereospecific PARP-1 Inhibitor Isoindolinone NMS-P515.
Journal: ACS medicinal chemistry letters
Published: November 22, 2018
Phase I dose escalation study of NMS-1286937, an orally available Polo-Like Kinase 1 inhibitor, in patients with advanced or metastatic solid tumors.
Journal: Investigational new drugs
Published: June 02, 2017
Afatinib Is a New Therapeutic Approach in Chordoma with a Unique Ability to Target EGFR and Brachyury.
Journal: Molecular cancer therapeutics
Published: April 12, 2017
Establishment and genomic characterization of the new chordoma cell line Chor-IN-1.
Journal: Scientific reports
Published: April 03, 2017
Discovery of Entrectinib: A New 3-Aminoindazole As a Potent Anaplastic Lymphoma Kinase (ALK), c-ros Oncogene 1 Kinase (ROS1), and Pan-Tropomyosin Receptor Kinases (Pan-TRKs) inhibitor.
Journal: Journal of medicinal chemistry
Published: March 23, 2016
Entrectinib, a Pan-TRK, ROS1, and ALK Inhibitor with Activity in Multiple Molecularly Defined Cancer Indications.
Journal: Molecular cancer therapeutics
Published: September 11, 2015
Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy.
Journal: Journal of medicinal chemistry
Published: July 30, 2015
Novel CAD-ALK gene rearrangement is drugable by entrectinib in colorectal cancer.
Journal: British journal of cancer
Published: July 17, 2015
Last Updated: 09/26/2026