Ayyiliath M. Sajith
Tumkur, KA 572107, India
Last Updated: 09/26/2026
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Found 17 publications
NMI-SO2Cl2-Mediated Amide Bond Formation: Facile Synthesis of Some Dihydrotriazolopyrimidine Amide Derivatives as Potential Anti-Inflammatory and Anti-Tubercular Agents.
Journal: Pharmaceuticals (Basel, Switzerland)
Published: November 21, 2023
Sub-pocket-focused designing of tacrine derivatives as potential acetylcholinesterase inhibitors.
Journal: Computers in biology and medicine
Published: December 01, 2022
Exploration of NMI-MsCl mediated amide bond formation for the synthesis of novel 3,5-substituted-1,2,4-oxadiazole derivatives: synthesis, evaluation of anti-inflammatory activity and molecular docking studies.
Journal: Molecular diversity
Published: March 21, 2022
Targeting NLRP3 signaling by a novel-designed sulfonylurea compound for inhibition of microglial inflammation.
Journal: Bioorganic & medicinal chemistry
Published: October 06, 2021
Design, synthesis and molecular docking studies of some 1-(5-(2-fluoro-5-(trifluoromethoxy)phenyl)-1,2,4-oxadiazol-3-yl)piperazine derivatives as potential anti-inflammatory agents.
Journal: Molecular diversity
Published: June 08, 2021
Application of NMI-TfCl-mediated amide bond formation in the synthesis of biologically relevant oxadiazole derivatives employing less basic (hetero)aryl amines.
Journal: Molecular diversity
Published: May 27, 2021
Pyrimidine-2,4-dione targets STAT3 signaling pathway to induce cytotoxicity in hepatocellular carcinoma cells.
Journal: Bioorganic & medicinal chemistry letters
Published: May 21, 2021
Epigenetic modulation and apoptotic induction by a novel imidazo-benzamide derivative in human lung adenocarcinoma cells.
Journal: Daru : journal of Faculty of Pharmacy, Tehran University of Medical Sciences
Published: March 30, 2021
Structural Optimization of 2,3-Dihydro-1H-cyclopenta[b]quinolines Targeting the Noncatalytic RVxF Site of Protein Phosphatase 1 for HIV-1 Inhibition.
Journal: ACS infectious diseases
Published: December 01, 2020
Drug Re-purposing Approach and Potential Therapeutic Strategies to Treat COVID-19.
Journal: Mini reviews in medicinal chemistry
Published: May 28, 2020
Design, synthesis, and screening of sulfonylurea-derived NLRP3 inflammasome inhibitors.
Journal: Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents
Published: July 19, 2019
Last Updated: 09/26/2026