Balazs Kramos

Budapest, BU 1103, Hungary

Last Updated: 09/26/2026

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Found 25 publications

The Discovery of RGH-706, a Highly Efficacious MCH1 Receptor Antagonist, for the Treatment of Obesity and Insatiable Hunger.

The Discovery of RGH-706, a Highly Efficacious MCH1 Receptor Antagonist, for the Treatment of Obesity and Insatiable Hunger.

Journal: Journal of medicinal chemistry
Published: January 22, 2026

Correction to "Discovery of an In Vitro and In Vivo Potent Nicotinic α7 Positive Allosteric Modulator Clinical Candidate Molecule (RGH-857)".

Correction to "Discovery of an In Vitro and In Vivo Potent Nicotinic α7 Positive Allosteric Modulator Clinical Candidate Molecule (RGH-857)".

Journal: Journal of medicinal chemistry
Published: January 19, 2026

Discovery of an In Vitro and In Vivo Potent Nicotinic α7 Positive Allosteric Modulator Clinical Candidate Molecule (RGH-857).

Discovery of an In Vitro and In Vivo Potent Nicotinic α7 Positive Allosteric Modulator Clinical Candidate Molecule (RGH-857).

Journal: Journal of medicinal chemistry
Published: December 29, 2025

Gymnopeptides C and D, Highly N-Methylated Fungal Cyclopeptides.

Gymnopeptides C and D, Highly N-Methylated Fungal Cyclopeptides.

Journal: Journal of natural products
Published: February 27, 2025

Ligand Binding and Functional Effect of Novel Bicyclic α5 GABAA Receptor Negative Allosteric Modulators.

Ligand Binding and Functional Effect of Novel Bicyclic α5 GABAA Receptor Negative Allosteric Modulators.

Journal: Journal of chemical information and modeling
Published: December 17, 2024

Development of dual V1a/V2 antagonists containing triazolobenzazepine scaffold.

Development of dual V1a/V2 antagonists containing triazolobenzazepine scaffold.

Journal: European journal of medicinal chemistry
Published: October 02, 2024

Novel-Type GABAB PAMs: Structure-Activity Relationship in Light of the Protein Structure.

Novel-Type GABAB PAMs: Structure-Activity Relationship in Light of the Protein Structure.

Journal: ACS medicinal chemistry letters
Published: December 20, 2023

Optimization of Novel α7 Nicotinic Acetylcholine Receptor Positive Allosteric Modulators and the Discovery of a Preclinical Development Candidate Molecule (RGH-560).

Optimization of Novel α7 Nicotinic Acetylcholine Receptor Positive Allosteric Modulators and the Discovery of a Preclinical Development Candidate Molecule (RGH-560).

Journal: Journal of medicinal chemistry
Published: November 21, 2023

Novel imidazo[1,5-a]quinoxaline derivatives: SAR, selectivity and modeling challenges en route to the identification of an α5-GABAA receptor NAM.

Novel imidazo[1,5-a]quinoxaline derivatives: SAR, selectivity and modeling challenges en route to the identification of an α5-GABAA receptor NAM.

Journal: Bioorganic & medicinal chemistry letters
Published: August 30, 2022

Potential Mechanisms for Why Not All Antipsychotics Are Able to Occupy Dopamine D3 Receptors in the Brain in vivo.

Potential Mechanisms for Why Not All Antipsychotics Are Able to Occupy Dopamine D3 Receptors in the Brain in vivo.

Journal: Frontiers in psychiatry
Published: September 29, 2021

Synthesis and Characterization of New V1A Antagonist Compounds: The Separation of Four Atropisomeric Stereoisomers.

Synthesis and Characterization of New V1A Antagonist Compounds: The Separation of Four Atropisomeric Stereoisomers.

Journal: Journal of medicinal chemistry
Published: July 13, 2021

HTS-based discovery and optimization of novel positive allosteric modulators of the α7 nicotinic acetylcholine receptor.

HTS-based discovery and optimization of novel positive allosteric modulators of the α7 nicotinic acetylcholine receptor.

Journal: European journal of medicinal chemistry
Published: February 26, 2021
Showing 1-12 of 25

Last Updated: 09/26/2026