Bohdan Waszkowycz

BioCity, Pennyfoot Street, U.K
Nottingham, ENG NG11GF, United Kingdom

Last Updated: 09/26/2026

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Found 18 publications

Development of Structurally Simplified, Non-azadecalin Glucocorticoid Antagonists which Demonstrate In Vivo Activity.

Development of Structurally Simplified, Non-azadecalin Glucocorticoid Antagonists which Demonstrate In Vivo Activity.

Journal: Journal of medicinal chemistry

Published: April 07, 2026

Discovery and Optimization of wt-RET/KDR-Selective Inhibitors of RETV804M Kinase.

Discovery and Optimization of wt-RET/KDR-Selective Inhibitors of RETV804M Kinase.

Journal: ACS medicinal chemistry letters

Published: December 17, 2019

Cell-Active Small Molecule Inhibitors of the DNA-Damage Repair Enzyme Poly(ADP-ribose) Glycohydrolase (PARG): Discovery and Optimization of Orally Bioavailable Quinazolinedione Sulfonamides.

Cell-Active Small Molecule Inhibitors of the DNA-Damage Repair Enzyme Poly(ADP-ribose) Glycohydrolase (PARG): Discovery and Optimization of Orally Bioavailable Quinazolinedione Sulfonamides.

Journal: Journal of medicinal chemistry

Published: November 08, 2018

Discovery and Optimization of Allosteric Inhibitors of Mutant Isocitrate Dehydrogenase 1 (R132H IDH1) Displaying Activity in Human Acute Myeloid Leukemia Cells.

Discovery and Optimization of Allosteric Inhibitors of Mutant Isocitrate Dehydrogenase 1 (R132H IDH1) Displaying Activity in Human Acute Myeloid Leukemia Cells.

Journal: Journal of medicinal chemistry

Published: December 23, 2016

Enhancer Activation by Pharmacologic Displacement of LSD1 from GFI1 Induces Differentiation in Acute Myeloid Leukemia.

Enhancer Activation by Pharmacologic Displacement of LSD1 from GFI1 Induces Differentiation in Acute Myeloid Leukemia.

Journal: Cell reports

Published: November 29, 2016

First-in-Class Chemical Probes against Poly(ADP-ribose) Glycohydrolase (PARG) Inhibit DNA Repair with Differential Pharmacology to Olaparib.

First-in-Class Chemical Probes against Poly(ADP-ribose) Glycohydrolase (PARG) Inhibit DNA Repair with Differential Pharmacology to Olaparib.

Journal: ACS chemical biology

Published: October 01, 2016

Identification of selective inhibitors of RET and comparison with current clinical candidates through development and validation of a robust screening cascade.

Identification of selective inhibitors of RET and comparison with current clinical candidates through development and validation of a robust screening cascade.

Journal: F1000Research

Published: July 19, 2016

Anilinoquinazoline inhibitors of the RET kinase domain-Elaboration of the 7-position.

Anilinoquinazoline inhibitors of the RET kinase domain-Elaboration of the 7-position.

Journal: Bioorganic & medicinal chemistry letters

Published: February 04, 2016

Application of virtual screening to the discovery of novel nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with potential for the treatment of cancer and axonopathies.

Application of virtual screening to the discovery of novel nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with potential for the treatment of cancer and axonopathies.

Journal: Bioorganic & medicinal chemistry letters

Published: February 02, 2016

The discovery of 2-substituted phenol quinazolines as potent RET kinase inhibitors with improved KDR selectivity.

The discovery of 2-substituted phenol quinazolines as potent RET kinase inhibitors with improved KDR selectivity.

Journal: European journal of medicinal chemistry

Published: August 27, 2015

A reversed sulfonamide series of selective RORc inverse agonists.

A reversed sulfonamide series of selective RORc inverse agonists.

Journal: Bioorganic & medicinal chemistry letters

Published: September 05, 2014

Toxoflavins and deazaflavins as the first reported selective small molecule inhibitors of tyrosyl-DNA phosphodiesterase II.

Toxoflavins and deazaflavins as the first reported selective small molecule inhibitors of tyrosyl-DNA phosphodiesterase II.

Journal: Journal of medicinal chemistry

Published: July 18, 2013

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Last Updated: 09/26/2026