Last Updated: 09/26/2026
Save publications for later
Sign Up
Not sure about your diagnosis?
Check Your Symptoms
Found 37 publications
Sample optimizations to enable the structure determination of biotin-dependent carboxylases.
Journal: Methods in enzymology
Published: November 21, 2024
Exploring monocyclic core: Discovery of pyrrol-2-one derivatives as a new series of potent MCHR1 antagonists with in vivo efficacy.
Journal: European journal of medicinal chemistry
Published: April 27, 2024
Development of BET Inhibitors as Potential Treatments for Cancer: Optimization of Pharmacokinetic Properties.
Journal: ACS medicinal chemistry letters
Published: July 21, 2022
Quantification of Linrodostat and its metabolites: Overcoming bioanalytical challenges in support of a discovery Indoleamine 2,3 dioxygenase program.
Journal: Journal of chromatography. B, Analytical technologies in the biomedical and life sciences
Published: December 14, 2021
Discovery and Preclinical Pharmacology of an Oral Bromodomain and Extra-Terminal (BET) Inhibitor Using Scaffold-Hopping and Structure-Guided Drug Design.
Journal: Journal of medicinal chemistry
Published: September 20, 2021
Conformational-Analysis-Guided Discovery of 2,3-Disubstituted Pyridine IDO1 Inhibitors.
Journal: ACS medicinal chemistry letters
Published: April 21, 2021
Development of BET inhibitors as potential treatments for cancer: A search for structural diversity.
Development of BET inhibitors as potential treatments for cancer: A search for structural diversity.
Journal: Bioorganic & medicinal chemistry letters
Published: March 12, 2021
Discovery of Imidazopyridines as Potent Inhibitors of Indoleamine 2,3-Dioxygenase 1 for Cancer Immunotherapy.
Journal: ACS medicinal chemistry letters
Published: January 12, 2021
Discovery and Preclinical Evaluation of BMS-986242, a Potent, Selective Inhibitor of Indoleamine-2,3-dioxygenase 1.
Journal: ACS medicinal chemistry letters
Published: December 20, 2020
Potent, Orally Bioavailable, and Efficacious Macrocyclic Inhibitors of Factor XIa. Discovery of Pyridine-Based Macrocycles Possessing Phenylazole Carboxamide P1 Groups.
Journal: Journal of medicinal chemistry
Published: December 14, 2019
Discovery of a Lead Triphenylethanamine Cholesterol Ester Transfer Protein (CETP) Inhibitor.
Journal: ACS medicinal chemistry letters
Published: March 04, 2019
Pharmacokinetics of 40 kDa PEG in rodents using high-field NMR spectroscopy.
Journal: Journal of pharmaceutical and biomedical analysis
Published: February 15, 2019
Last Updated: 09/26/2026