Last Updated: 09/26/2026
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Found 24 publications
GIPR gene expression in testis is mouse specific and can impact male mouse fertility.
Journal: Andrology
Published: October 22, 2021
GIPR antagonist antibodies conjugated to GLP-1 peptide are bispecific molecules that decrease weight in obese mice and monkeys.
Journal: Cell reports. Medicine
Published: April 23, 2020
Chronic glucose-dependent insulinotropic polypeptide receptor (GIPR) agonism desensitizes adipocyte GIPR activity mimicking functional GIPR antagonism.
Journal: Nature communications
Published: September 18, 2019
Anti-obesity effects of GIPR antagonists alone and in combination with GLP-1R agonists in preclinical models.
Journal: Science translational medicine
Published: February 16, 2018
Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disrupters of Glucokinase-Glucokinase Regulatory Protein (GK-GKRP) Binding: Strategic Use of a N → S (nN → σ*S-X) Interaction for Conformational Constraint.
Journal: Journal of medicinal chemistry
Published: November 10, 2015
Haploinsufficiency of the Insulin Receptor in the Presence of a Splice-Site Mutation in Ppp2r2a Results in a Novel Digenic Mouse Model of Type 2 Diabetes.
Journal: Diabetes
Published: September 10, 2015
Small Molecule Disruptors of the Glucokinase-Glucokinase Regulatory Protein Interaction: 5. A Novel Aryl Sulfone Series, Optimization Through Conformational Analysis.
Journal: Journal of medicinal chemistry
Published: April 28, 2015
Pharmacologic Effects of FGF21 Are Independent of the "Browning" of White Adipose Tissue.
Journal: Cell metabolism
Published: November 13, 2014
Molecular targeting of the GK-GKRP pathway in diabetes.
Journal: Expert opinion on therapeutic targets
Published: October 18, 2014
A mutation in Ampd2 is associated with nephrotic syndrome and hypercholesterolemia in mice.
Journal: Lipids in health and disease
Published: July 21, 2014
Last Updated: 09/26/2026