Djordje Musil

Frankfurter Str. 250
Darmstadt, HE 64293, Germany

Last Updated: 09/26/2026

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Found 39 publications

Discovery of ART5537: A Potent and Selective Small-Molecule Probe for EXO1.

Discovery of ART5537: A Potent and Selective Small-Molecule Probe for EXO1.

Journal: Journal of medicinal chemistry

Published: December 08, 2025

Phenotypic Hit Identification and Optimization of Novel Pan-TEAD and Subtype-Selective Inhibitors.

Phenotypic Hit Identification and Optimization of Novel Pan-TEAD and Subtype-Selective Inhibitors.

Journal: Journal of medicinal chemistry

Published: November 10, 2025

Phenotypic Hit Identification and Optimization of Novel Pan-TEAD and Subtype-Selective Inhibitors.

Phenotypic Hit Identification and Optimization of Novel Pan-TEAD and Subtype-Selective Inhibitors.

Journal: Journal of medicinal chemistry

Published: November 10, 2025

Pushing the limits of hydrogen/deuterium exchange mass spectrometry to study protein:fragment low affinity interactions.

Pushing the limits of hydrogen/deuterium exchange mass spectrometry to study protein:fragment low affinity interactions.

Journal: Communications chemistry

Published: October 03, 2025

MoA Studies of the TEAD P-Site Binding Ligand MSC-4106 and Its Optimization to TEAD1-Selective Amide M3686.

MoA Studies of the TEAD P-Site Binding Ligand MSC-4106 and Its Optimization to TEAD1-Selective Amide M3686.

Journal: Journal of medicinal chemistry

Published: December 20, 2024

Discovery of reversible and covalent TEAD 1 selective inhibitors MSC-1254 and MSC-5046 based on one scaffold.

Discovery of reversible and covalent TEAD 1 selective inhibitors MSC-1254 and MSC-5046 based on one scaffold.

Journal: Bioorganic & medicinal chemistry letters

Published: July 21, 2024

On the humanization of VHHs: Prospective case studies, experimental and computational characterization of structural determinants for functionality.

On the humanization of VHHs: Prospective case studies, experimental and computational characterization of structural determinants for functionality.

Journal: Protein science : a publication of the Protein Society

Published: July 04, 2024

Discovery of Cycloalkyl[c]thiophenes as Novel Scaffolds for Hypoxia-Inducible Factor-2α Inhibitors.

Discovery of Cycloalkyl[c]thiophenes as Novel Scaffolds for Hypoxia-Inducible Factor-2α Inhibitors.

Journal: Journal of medicinal chemistry

Published: July 05, 2023

Discovery of quinazoline HPK1 inhibitors with high cellular potency.

Discovery of quinazoline HPK1 inhibitors with high cellular potency.

Journal: Bioorganic & medicinal chemistry

Published: February 23, 2023

Selective Wee1 Inhibitors Led to Antitumor Activity In Vitro and Correlated with Myelosuppression.

Selective Wee1 Inhibitors Led to Antitumor Activity In Vitro and Correlated with Myelosuppression.

Journal: ACS medicinal chemistry letters

Published: November 11, 2022

Optimization of TEAD P-Site Binding Fragment Hit into In Vivo Active Lead MSC-4106.

Optimization of TEAD P-Site Binding Fragment Hit into In Vivo Active Lead MSC-4106.

Journal: Journal of medicinal chemistry

Published: June 28, 2022

Optimization of a Screening Hit toward M2912, an Oral Tankyrase Inhibitor with Antitumor Activity in Colorectal Cancer Models.

Optimization of a Screening Hit toward M2912, an Oral Tankyrase Inhibitor with Antitumor Activity in Colorectal Cancer Models.

Journal: Journal of medicinal chemistry

Published: July 13, 2021

Showing 1-12 of 39

Last Updated: 09/26/2026