Erik De Heuvel
Amsterdam, NH 1081HZ, Netherlands
Last Updated: 09/26/2026
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Found 10 publications
To Target or Not to Target Schistosoma mansoni Cyclic Nucleotide Phosphodiesterase 4A?
Journal: International journal of molecular sciences
Published: February 07, 2023
Discovery of Diaryl Ether Substituted Tetrahydrophthalazinones as TbrPDEB1 Inhibitors Following Structure-Based Virtual Screening.
Journal: Frontiers in chemistry
Published: September 18, 2020
Identification of Phenylphthalazinones as a New Class of Leishmania infantum Inhibitors.
Journal: ChemMedChem
Published: September 20, 2019
Evaluation of phthalazinone phosphodiesterase inhibitors with improved activity and selectivity against Trypanosoma cruzi.
Journal: The Journal of antimicrobial chemotherapy
Published: July 19, 2019
Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors (Part 2).
Journal: Bioorganic & medicinal chemistry
Published: May 11, 2019
Stable pantothenamide bioisosteres: novel antibiotics for Gram-positive bacteria.
Journal: The Journal of antibiotics
Published: February 15, 2019
Screening of a PDE-focused library identifies imidazoles with in vitro and in vivo antischistosomal activity.
Journal: International journal for parasitology. Drugs and drug resistance
Published: November 15, 2018
Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors.
Journal: Bioorganic & medicinal chemistry
Published: September 17, 2018
Targeting a Subpocket in Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1) Enables the Structure-Based Discovery of Selective Inhibitors with Trypanocidal Activity.
Journal: Journal of medicinal chemistry
Published: April 20, 2018
Discovery of small molecule vanin inhibitors: new tools to study metabolism and disease.
Journal: ACS chemical biology
Published: December 29, 2012
Showing 1-10 of 10
Last Updated: 09/26/2026