Eva Tloustova

Prague, PR 16610, Czech Republic

Last Updated: 09/26/2026

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Found 25 publications

On-Resin Assembly of Macrocyclic Inhibitors of Cryptococcus neoformans May1: A Pathway to Potent Antifungal Agents.

On-Resin Assembly of Macrocyclic Inhibitors of Cryptococcus neoformans May1: A Pathway to Potent Antifungal Agents.

Journal: Journal of medicinal chemistry

Published: April 22, 2025

Sulfonated Hydroxyaryl-Tetrazines with Increased pKa for Accelerated Bioorthogonal Click-to-Release Reactions in Cells.

Sulfonated Hydroxyaryl-Tetrazines with Increased pKa for Accelerated Bioorthogonal Click-to-Release Reactions in Cells.

Journal: Angewandte Chemie (International ed. in English)

Published: June 21, 2024

Structure-Based Drug Design of ADRA2A Antagonists Derived from Yohimbine.

Structure-Based Drug Design of ADRA2A Antagonists Derived from Yohimbine.

Journal: Journal of medicinal chemistry

Published: June 10, 2024

Discovery of a potent and selective human AC2 inhibitor based on 7-deazapurine analogues of adefovir.

Discovery of a potent and selective human AC2 inhibitor based on 7-deazapurine analogues of adefovir.

Journal: Bioorganic & medicinal chemistry

Published: July 28, 2023

Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors.

Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors.

Journal: Journal of medicinal chemistry

Published: May 03, 2023

Synthesis and anti-trypanosomal evaluation of novel N-branched acyclic nucleoside phosphonates bearing 7-aryl-7-deazapurine nucleobase.

Synthesis and anti-trypanosomal evaluation of novel N-branched acyclic nucleoside phosphonates bearing 7-aryl-7-deazapurine nucleobase.

Journal: European journal of medicinal chemistry

Published: May 03, 2022

Halogen-Dance-Based Synthesis of Phosphonomethoxyethyl (PME) Substituted 2-Aminothiazoles as Potent Inhibitors of Bacterial Adenylate Cyclases.

Halogen-Dance-Based Synthesis of Phosphonomethoxyethyl (PME) Substituted 2-Aminothiazoles as Potent Inhibitors of Bacterial Adenylate Cyclases.

Journal: ChemMedChem

Published: August 24, 2021

Re-emerging Aspartic Protease Targets: Examining Cryptococcus neoformans Major Aspartyl Peptidase 1 as a Target for Antifungal Drug Discovery.

Re-emerging Aspartic Protease Targets: Examining Cryptococcus neoformans Major Aspartyl Peptidase 1 as a Target for Antifungal Drug Discovery.

Journal: Journal of medicinal chemistry

Published: May 19, 2021

Synthesis and Antitrypanosomal Activity of 6-Substituted 7-Methyl-7-deazapurine Nucleosides.

Synthesis and Antitrypanosomal Activity of 6-Substituted 7-Methyl-7-deazapurine Nucleosides.

Journal: ACS infectious diseases

Published: March 26, 2021

Synthesis and anti-trypanosomal activity of 3'-fluororibonucleosides derived from 7-deazapurine nucleosides.

Synthesis and anti-trypanosomal activity of 3'-fluororibonucleosides derived from 7-deazapurine nucleosides.

Journal: Bioorganic & medicinal chemistry letters

Published: February 04, 2021

Acyclic nucleoside phosphonates with 2-aminothiazole base as inhibitors of bacterial and mammalian adenylate cyclases.

Acyclic nucleoside phosphonates with 2-aminothiazole base as inhibitors of bacterial and mammalian adenylate cyclases.

Journal: European journal of medicinal chemistry

Published: November 24, 2020

Synthesis and Cytotoxic and Antiviral Activity Profiling of All-Four Isomeric Series of Pyrido-Fused 7-Deazapurine Ribonucleosides.

Synthesis and Cytotoxic and Antiviral Activity Profiling of All-Four Isomeric Series of Pyrido-Fused 7-Deazapurine Ribonucleosides.

Journal: Chemistry (Weinheim an der Bergstrasse, Germany)

Published: March 04, 2020

Showing 1-12 of 25

Last Updated: 09/26/2026