Francis Giraud
Clermont-ferrand, 63000, France
Last Updated: 09/26/2026
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Found 26 publications
Recent developments in Haspin kinase inhibitors: Structure, synthesis and activities.
Journal: Bioorganic & medicinal chemistry
Published: March 03, 2026
Synthesis of 1H-Pyrrolo[3,2-g]isoquinoline Derivatives as Ligands Targeting Haspin Kinase.
Journal: Molecules (Basel, Switzerland)
Published: September 26, 2025
Synthesis and biological activity of 1H-pyrrolo[3,2-g]isoquinolines as Haspin kinase inhibitors.
Journal: Bioorganic & medicinal chemistry
Published: December 02, 2024
Liposomes loaded with daunorubicin and an emetine prodrug for improved selective cytotoxicity towards acute myeloid leukaemia cells.
Journal: International journal of pharmaceutics
Published: June 07, 2024
Synthesis of diversely substituted pyridin-2(1H)-ones and in vivo evaluation of their anti-allodynic effect on cutaneous inflammatory mechanical allodynia.
Journal: RSC medicinal chemistry
Published: May 22, 2024
The Nitro Group Reshapes the Effects of Pyrido[3,4-g]quinazoline Derivatives on DYRK/CLK Activity and RNA Splicing in Glioblastoma Cells.
Journal: Cancers
Published: December 30, 2023
Synthesis and biological evaluation of 1H-pyrrolo[3,2-g]isoquinolines.
Journal: Bioorganic & medicinal chemistry
Published: December 22, 2023
Synthesis, kinase inhibition and anti-leukemic activities of diversely substituted indolopyrazolocarbazoles.
Journal: European journal of medicinal chemistry
Published: December 20, 2023
Synthesis and Kinase Inhibitory Potencies of Pyrazolo[3,4-g]isoquinolines.
Journal: Molecules (Basel, Switzerland)
Published: July 18, 2022
Synthesis of new pyrazolo[4,3-a]phenanthridine Pim-1 inhibitors and evaluation of their cytotoxic activity towards the MOLM-13 acute myeloid leukemia cell line.
Journal: Bioorganic & medicinal chemistry letters
Published: June 07, 2022
Synthesis and biological evaluation of Haspin inhibitors: Kinase inhibitory potency and cellular activity.
Journal: European journal of medicinal chemistry
Published: March 15, 2022
Last Updated: 09/26/2026