Fredrik Bjorkling
Copenhagen, Denmark
Last Updated: 09/26/2026
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Found 24 publications
Pyridine indole hybrids as novel potent CYP17A1 inhibitors.
Journal: Journal of enzyme inhibition and medicinal chemistry
Published: February 14, 2025
Polymyxins with Potent Antibacterial Activity against Colistin-Resistant Pathogens: Fine-Tuning Hydrophobicity with Unnatural Amino Acids.
Journal: Journal of medicinal chemistry
Published: January 03, 2024
Studies of antibacterial activity (in vitro and in vivo) and mode of action for des-acyl tridecaptins (DATs).
Journal: European journal of medicinal chemistry
Published: November 09, 2023
Exploring the Potential of Sulfur Moieties in Compounds Inhibiting Steroidogenesis.
Journal: Biomolecules
Published: July 31, 2023
Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues.
Journal: Bioorganic chemistry
Published: July 26, 2023
Non-steroidal CYP17A1 Inhibitors: Discovery and Assessment.
Journal: Journal of medicinal chemistry
Published: May 16, 2023
Antimicrobial Peptides Incorporating Halogenated Marine-Derived Amino Acid Substituents.
Journal: ACS medicinal chemistry letters
Published: March 15, 2023
Selected strategies to fight pathogenic bacteria.
Journal: Journal of enzyme inhibition and medicinal chemistry
Published: January 11, 2023
Correction to "Structural Basis of Metallo-β-lactamase Inhibition by N-Sulfamoylpyrrole-2-carboxylates".
Journal: ACS infectious diseases
Published: October 04, 2021
Peptide/β-Peptoid Hybrids with Ultrashort PEG-Like Moieties: Effects on Hydrophobicity, Antibacterial Activity and Hemolytic Properties.
Journal: International journal of molecular sciences
Published: June 01, 2021
Structural Basis of Metallo-β-lactamase Inhibition by N-Sulfamoylpyrrole-2-carboxylates.
Journal: ACS infectious diseases
Published: May 18, 2021
Last Updated: 09/26/2026