Giada Cernicchi
Perugia, Italy
Last Updated: 09/26/2026
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Found 10 publications
2-Phenylquinolines Exhibit Anti-Severe Acute Respiratory Syndrome Coronavirus-2 Activity Through the Nonstructural Protein 13 Helicase Inhibition.
Journal: ChemMedChem
Published: November 21, 2025
In Vitro and In Vivo Investigations into the Potential of Quinazoline and Quinoline Derivatives as NorA Efflux Pump Inhibitors Against Resistant Staphylococcus aureus Strains.
Journal: Antibiotics (Basel, Switzerland)
Published: February 14, 2025
NorA Efflux Pump Inhibitors: Expanding SAR Knowledge of Pyrazolo[4,3-c][1,2]benzothiazine 5,5-Dioxide Derivatives.
Journal: Archiv der Pharmazie
Published: December 12, 2024
Addressing Data Point Homogeneity and Annotation Challenges to Enhance Data-Driven Approaches: The S. aureus NorA Efflux Pump Case Study.
Journal: ChemMedChem
Published: November 16, 2024
Discovery of 2-phenylquinazolines as potent Mycobacterium avium efflux pump inhibitors able to synergize with clarithromycin against clinical isolate.
Journal: Archiv der Pharmazie
Published: April 19, 2024
Inhibition of Staphylococcus pseudintermedius Efflux Pumps by Using Staphylococcus aureus NorA Efflux Pump Inhibitors.
Journal: Antibiotics (Basel, Switzerland)
Published: March 24, 2023
New C-6 functionalized quinoline NorA inhibitors strongly synergize with ciprofloxacin against planktonic and biofilm growing resistant Staphylococcus aureus strains.
Journal: European journal of medicinal chemistry
Published: May 30, 2022
Discovery of 2-Phenylquinolines with Broad-Spectrum Anti-coronavirus Activity.
Journal: ACS medicinal chemistry letters
Published: March 18, 2022
Microbial Efflux Pump Inhibitors: A Journey around Quinoline and Indole Derivatives.
Journal: Molecules (Basel, Switzerland)
Published: October 11, 2021
From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search.
Journal: ChemMedChem
Published: April 23, 2021
Showing 1-10 of 10
Last Updated: 09/26/2026