Giulia Caron
Via Quarello15
Turin, 10135, Italy
Turin, 10135, Italy
Last Updated: 09/26/2026
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Found 75 publications
MK4 Repositioning for IAHSP: Overcoming In Vivo Data Gaps through In Silico Refinement and In Vitro Validation.
Journal: ACS chemical neuroscience
Published: February 09, 2026
SangsterLogP - the largest publicly available dataset of logP values.
Journal: Scientific data
Published: January 14, 2026
BBB-Permeable PROTACs: Where Do We Stand?
Journal: ACS medicinal chemistry letters
Published: December 22, 2025
Bellerophon: An Automated Tool for PROTAC Decomposition.
Journal: ACS medicinal chemistry letters
Published: December 22, 2025
Massive barcode-free chemical screenings enable the discovery of bioactive macrocycles with passive membrane permeability.
Journal: Nature communications
Published: December 17, 2025
Linker Methylation as a Strategy to Enhance PROTAC Oral Bioavailability: Insights from Molecular Properties and Conformational Analysis.
Journal: Journal of medicinal chemistry
Published: August 01, 2025
Smart Integration of Structural Biology and Medicinal Chemistry to Unlock Target-Driven Drug Discovery.
Journal: Medicinal research reviews
Published: April 23, 2025
Finding a needle in the haystack: ADME and pharmacokinetics/pharmacodynamics characterization and optimization toward orally available bifunctional protein degraders.
Journal: Expert opinion on drug discovery
Published: February 16, 2025
Macrocyclization: Enhancing Drug-like Properties of Discoidin Domain Receptor Kinase Inhibitors.
Journal: ACS medicinal chemistry letters
Published: December 19, 2024
Restoring adapter protein complex 4 function with small molecules: an in silico approach to spastic paraplegia 50.
Journal: Protein science : a publication of the Protein Society
Published: August 03, 2024
IMHB-Mediated Chameleonicity in Drug Design: A Focus on Structurally Related PROTACs.
Journal: Journal of medicinal chemistry
Published: June 29, 2024
Molecular properties, including chameleonicity, as essential tools for designing the next generation of oral beyond rule of five drugs.
Journal: ADMET & DMPK
Published: March 22, 2024
Last Updated: 09/26/2026