Giusy Tassone

Via A. Moro 2
Siena, 53100, Italy

Last Updated: 09/26/2026

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Found 27 publications

Morita-Baylis-Hillman Adduct Chemistry as a Tool for the Design of Lysine-Targeted Covalent Ligands.

Morita-Baylis-Hillman Adduct Chemistry as a Tool for the Design of Lysine-Targeted Covalent Ligands.

Journal: ACS medicinal chemistry letters
Published: October 01, 2024

Metal Ion Binding to Human Glutaminyl Cyclase: A Structural Perspective.

Metal Ion Binding to Human Glutaminyl Cyclase: A Structural Perspective.

Journal: International journal of molecular sciences
Published: July 02, 2024

Exploiting the bile acid binding protein as transporter of a Cholic Acid/Mirin bioconjugate for potential applications in liver cancer therapy.

Exploiting the bile acid binding protein as transporter of a Cholic Acid/Mirin bioconjugate for potential applications in liver cancer therapy.

Journal: Scientific reports
Published: June 21, 2024

A Facile Access to Green Fluorescent Albumin Derivatives.

A Facile Access to Green Fluorescent Albumin Derivatives.

Journal: Chembiochem : a European journal of chemical biology
Published: December 22, 2023

The discovery of aryl-2-nitroethyl triamino pyrimidines as anti-Trypanosoma brucei agents.

The discovery of aryl-2-nitroethyl triamino pyrimidines as anti-Trypanosoma brucei agents.

Journal: European journal of medicinal chemistry
Published: September 11, 2023

Antitarget, Anti-SARS-CoV-2 Leads, Drugs, and the Drug Discovery-Genetics Alliance Perspective.

Antitarget, Anti-SARS-CoV-2 Leads, Drugs, and the Drug Discovery-Genetics Alliance Perspective.

Journal: Journal of medicinal chemistry
Published: March 01, 2023

Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates.

Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates.

Journal: Journal of medicinal chemistry
Published: November 30, 2022

Exploiting ELIOT for Scaffold-Repurposing Opportunities: TRIM33 a Possible Novel E3 Ligase to Expand the Toolbox for PROTAC Design.

Exploiting ELIOT for Scaffold-Repurposing Opportunities: TRIM33 a Possible Novel E3 Ligase to Expand the Toolbox for PROTAC Design.

Journal: International journal of molecular sciences
Published: October 26, 2022

Structural Basis of Parasitic HSP90 ATPase Inhibition by Small Molecules.

Structural Basis of Parasitic HSP90 ATPase Inhibition by Small Molecules.

Journal: Pharmaceuticals (Basel, Switzerland)
Published: September 23, 2022

Structural Characterization of Human Heat Shock Protein 90 N-Terminal Domain and Its Variants K112R and K112A in Complex with a Potent 1,2,3-Triazole-Based Inhibitor.

Structural Characterization of Human Heat Shock Protein 90 N-Terminal Domain and Its Variants K112R and K112A in Complex with a Potent 1,2,3-Triazole-Based Inhibitor.

Journal: International journal of molecular sciences
Published: July 22, 2022

Dimerization of the C-type lectin-like receptor CD93 promotes its binding to Multimerin-2 in endothelial cells.

Dimerization of the C-type lectin-like receptor CD93 promotes its binding to Multimerin-2 in endothelial cells.

Journal: International journal of biological macromolecules
Published: July 15, 2022

1,2,4-Triazole-3-Thione Analogues with a 2-Ethylbenzoic Acid at Position 4 as VIM-type Metallo-β-Lactamase Inhibitors.

1,2,4-Triazole-3-Thione Analogues with a 2-Ethylbenzoic Acid at Position 4 as VIM-type Metallo-β-Lactamase Inhibitors.

Journal: ChemMedChem
Published: November 05, 2021
Showing 1-12 of 27

Last Updated: 09/26/2026