Last Updated: 09/26/2026
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Found 4 publications
A small molecule inhibitor of PCSK9 that antagonizes LDL receptor binding via interaction with a cryptic PCSK9 binding groove.
Journal: Bioorganic & medicinal chemistry
Published: August 23, 2019
Discovery and in vivo evaluation of alcohol-containing benzothiazoles as potent dual-targeting bacterial DNA supercoiling inhibitors.
Journal: Bioorganic & medicinal chemistry letters
Published: May 16, 2014
Design, synthesis and biological evaluation of α-substituted isonipecotic acid benzothiazole analogues as potent bacterial type II topoisomerase inhibitors.
Journal: Bioorganic & medicinal chemistry letters
Published: June 25, 2013
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Last Updated: 09/26/2026