Kasim A. Mookhtiar

Bengaluru, KA 560058, India

Last Updated: 09/26/2026

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Found 15 publications

Design and synthesis of novel spirocyclic carboxylic acids as potent and orally bioavailable DGAT1 inhibitors and their biological evaluation.

Design and synthesis of novel spirocyclic carboxylic acids as potent and orally bioavailable DGAT1 inhibitors and their biological evaluation.

Journal: Bioorganic & medicinal chemistry letters

Published: December 08, 2021

Recombinant irisin induces weight loss in high fat DIO mice through increase in energy consumption and thermogenesis.

Recombinant irisin induces weight loss in high fat DIO mice through increase in energy consumption and thermogenesis.

Journal: Biochemical and biophysical research communications

Published: August 13, 2019

Discovery and pharmacological evaluation of indole derivatives as potent and selective RORγt inverse agonist for multiple autoimmune conditions.

Discovery and pharmacological evaluation of indole derivatives as potent and selective RORγt inverse agonist for multiple autoimmune conditions.

Journal: Bioorganic & medicinal chemistry letters

Published: April 22, 2019

Discovery and evaluation of novel FAAH inhibitors in neuropathic pain model.

Discovery and evaluation of novel FAAH inhibitors in neuropathic pain model.

Journal: Bioorganic & medicinal chemistry letters

Published: October 08, 2018

Evaluation of separate role of intestine and liver in first pass metabolism of budesonide in rat.

Evaluation of separate role of intestine and liver in first pass metabolism of budesonide in rat.

Journal: Xenobiotica; the fate of foreign compounds in biological systems

Published: November 23, 2017

Modifications of flexible nonyl chain and nucleobase head group of (+)-erythro-9-(2's-hydroxy-3's-nonyl)adenine [(+)-EHNA] as adenosine deaminase inhibitors.

Modifications of flexible nonyl chain and nucleobase head group of (+)-erythro-9-(2's-hydroxy-3's-nonyl)adenine [(+)-EHNA] as adenosine deaminase inhibitors.

Journal: Bioorganic & medicinal chemistry

Published: April 24, 2017

Discovery of Potent and Selective A2A Antagonists with Efficacy in Animal Models of Parkinson's Disease and Depression.

Discovery of Potent and Selective A2A Antagonists with Efficacy in Animal Models of Parkinson's Disease and Depression.

Journal: ACS medicinal chemistry letters

Published: April 22, 2017

Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A2A Receptor Antagonists and Their Biological Evaluation.

Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A2A Receptor Antagonists and Their Biological Evaluation.

Journal: Journal of medicinal chemistry

Published: January 06, 2017

Discovery of liver-directed glucokinase activator having anti-hyperglycemic effect without hypoglycemia.

Discovery of liver-directed glucokinase activator having anti-hyperglycemic effect without hypoglycemia.

Journal: European journal of medicinal chemistry

Published: December 26, 2016

Discovery and evaluation of 1H-pyrrolo[2,3-b]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis.

Discovery and evaluation of 1H-pyrrolo[2,3-b]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis.

Journal: Bioorganic & medicinal chemistry letters

Published: December 13, 2016

Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A1 receptor antagonists and their biological evaluation.

Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A1 receptor antagonists and their biological evaluation.

Journal: Bioorganic & medicinal chemistry

Published: November 16, 2016

Design and synthesis of novel xanthine derivatives as potent and selective A2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases.

Design and synthesis of novel xanthine derivatives as potent and selective A2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases.

Journal: European journal of medicinal chemistry

Published: November 15, 2016

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Last Updated: 09/26/2026