Leandro A. Avelar-Alves
Duesseldorf, NW 40225, Germany
Last Updated: 09/26/2026
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Found 16 publications
Deciphering the Therapeutic Potential of Novel Pentyloxyamide-Based Class I, IIb HDAC Inhibitors against Therapy-Resistant Leukemia.
Journal: Journal of medicinal chemistry
Published: November 27, 2024
Characterization of the dehydrogenase-reductase DHRS2 and its involvement in histone deacetylase inhibition in urological malignancies.
Journal: Experimental cell research
Published: January 23, 2024
Activity of alkoxyamide-based histone deacetylase inhibitors against Plasmodium falciparum malaria parasites.
Journal: Experimental parasitology
Published: December 14, 2023
Over 40 Years of Fosmidomycin Drug Research: A Comprehensive Review and Future Opportunities.
Journal: Pharmaceuticals (Basel, Switzerland)
Published: October 28, 2022
Establishment and Evaluation of Dual HDAC/BET Inhibitors as Therapeutic Options for Germ Cell Tumors and Other Urological Malignancies.
Journal: Molecular cancer therapeutics
Published: March 24, 2022
Antiproliferation and Antiencystation Effect of Class II Histone Deacetylase Inhibitors on Acanthamoeba castellanii.
Journal: ACS infectious diseases
Published: January 07, 2022
Designing HDAC-PROTACs: lessons learned so far.
Journal: Future medicinal chemistry
Published: December 24, 2021
A short overview of resistance to approved histone deacetylase inhibitors.
Journal: Future medicinal chemistry
Published: May 07, 2021
Synergistic induction of apoptosis in resistant head and neck carcinoma and leukemia by alkoxyamide-based histone deacetylase inhibitors.
Journal: European journal of medicinal chemistry
Published: October 01, 2020
Structure-based design of selective histone deacetylase 6 zinc binding groups.
Journal: Journal of biomolecular structure & dynamics
Published: August 07, 2019
Novel reverse thia-analogs of fosmidomycin: Synthesis and antiplasmodial activity.
Journal: European journal of medicinal chemistry
Published: June 07, 2019
Recent advances in class IIa histone deacetylases research.
Journal: Bioorganic & medicinal chemistry
Published: March 29, 2019
Last Updated: 09/26/2026