Leopold Thabault

Brussels, BRU 1200, Belgium

Last Updated: 09/26/2026

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Found 12 publications

Olaparib Is a Mitochondrial Complex I Inhibitor That Kills Temozolomide-Resistant Human Glioblastoma Cells.

Olaparib Is a Mitochondrial Complex I Inhibitor That Kills Temozolomide-Resistant Human Glioblastoma Cells.

Journal: International journal of molecular sciences

Published: September 21, 2021

Correction to "Rational Design of Original Fused-Cycle Selective Inhibitors of Tryptophan 2,3-Dioxygenase".

Correction to "Rational Design of Original Fused-Cycle Selective Inhibitors of Tryptophan 2,3-Dioxygenase".

Journal: Journal of medicinal chemistry

Published: August 26, 2021

Rational Design of Original Fused-Cycle Selective Inhibitors of Tryptophan 2,3-Dioxygenase.

Rational Design of Original Fused-Cycle Selective Inhibitors of Tryptophan 2,3-Dioxygenase.

Journal: Journal of medicinal chemistry

Published: August 02, 2021

Investigation of chalcogen bioisosteric replacement in a series of heterocyclic inhibitors of tryptophan 2,3-dioxygenase.

Investigation of chalcogen bioisosteric replacement in a series of heterocyclic inhibitors of tryptophan 2,3-dioxygenase.

Journal: European journal of medicinal chemistry

Published: July 09, 2021

Discovery of small molecules interacting at lactate dehydrogenases tetrameric interface using a biophysical screening cascade.

Discovery of small molecules interacting at lactate dehydrogenases tetrameric interface using a biophysical screening cascade.

Journal: European journal of medicinal chemistry

Published: June 12, 2021

The metalloprotein YhcH is an anomerase providing N-acetylneuraminate aldolase with the open form of its substrate.

The metalloprotein YhcH is an anomerase providing N-acetylneuraminate aldolase with the open form of its substrate.

Journal: The Journal of biological chemistry

Published: February 23, 2021

Discovery of a novel lactate dehydrogenase tetramerization domain using epitope mapping and peptides.

Discovery of a novel lactate dehydrogenase tetramerization domain using epitope mapping and peptides.

Journal: The Journal of biological chemistry

Published: January 05, 2021

Unravelling the Allosteric Targeting of PHGDH at the ACT-Binding Domain with a Photoactivatable Diazirine Probe and Mass Spectrometry Experiments.

Unravelling the Allosteric Targeting of PHGDH at the ACT-Binding Domain with a Photoactivatable Diazirine Probe and Mass Spectrometry Experiments.

Journal: Molecules (Basel, Switzerland)

Published: December 31, 2020

Targeting protein self-association in drug design.

Targeting protein self-association in drug design.

Journal: Drug discovery today

Published: June 16, 2020

Interrogating the Lactate Dehydrogenase Tetramerization Site Using (Stapled) Peptides.

Interrogating the Lactate Dehydrogenase Tetramerization Site Using (Stapled) Peptides.

Journal: Journal of medicinal chemistry

Published: April 07, 2020

The putative Escherichia coli dehydrogenase YjhC metabolises two dehydrated forms of N-acetylneuraminate produced by some sialidases.

The putative Escherichia coli dehydrogenase YjhC metabolises two dehydrated forms of N-acetylneuraminate produced by some sialidases.

Journal: Bioscience reports

Published: March 25, 2020

1-(2-Hydroxybenzoyl)-thiosemicarbazides are promising antimicrobial agents targeting d-alanine-d-alanine ligase in bacterio.

1-(2-Hydroxybenzoyl)-thiosemicarbazides are promising antimicrobial agents targeting d-alanine-d-alanine ligase in bacterio.

Journal: European journal of medicinal chemistry

Published: May 04, 2018

Showing 1-12 of 12

Last Updated: 09/26/2026