Lisbeth Elster
Horsholm, 2970, Denmark
Last Updated: 09/26/2026
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Found 11 publications
Machine-Learning-Guided Peptide Drug Discovery: Development of GLP-1 Receptor Agonists with Improved Drug Properties.
Journal: Journal of medicinal chemistry
Published: July 08, 2024
Uncovering CNS access of lipidated exendin-4 analogues by quantitative whole-brain 3D light sheet imaging.
Journal: Neuropharmacology
Published: December 30, 2022
Half-Life Extending Modifications of Peptide YY3-36 Direct Receptor-Mediated Internalization.
Journal: Molecular pharmaceutics
Published: July 17, 2019
The identification of GPR3 inverse agonist AF64394; the first small molecule inhibitor of GPR3 receptor function.
Journal: Bioorganic & medicinal chemistry letters
Published: September 11, 2014
Optimisation of in silico derived 2-aminobenzimidazole hits as unprecedented selective kappa opioid receptor agonists.
Journal: Bioorganic & medicinal chemistry letters
Published: September 03, 2014
Structural basis for constitutive activity and agonist-induced activation of the enteroendocrine fat sensor GPR119.
Journal: British journal of pharmacology
Published: March 31, 2014
Design and optimization of quinazoline derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists: part 2.
Journal: Bioorganic & medicinal chemistry letters
Published: January 22, 2012
Design and optimization of quinazoline derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists.
Journal: Bioorganic & medicinal chemistry letters
Published: January 10, 2012
Showing 1-11 of 11
Last Updated: 09/26/2026