Lucas B. Hoelz

Pinheiral, RJ 27197000, Brazil

Last Updated: 09/26/2026

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Found 13 publications

Ponatinib: A Review of the History of Medicinal Chemistry behind Its Development.

Ponatinib: A Review of the History of Medicinal Chemistry behind Its Development.

Journal: Pharmaceuticals (Basel, Switzerland)

Published: August 15, 2024

A Selective Adenylyl Cyclase 1 Inhibitor Relieves Pain Without Causing Tolerance.

A Selective Adenylyl Cyclase 1 Inhibitor Relieves Pain Without Causing Tolerance.

Journal: Frontiers in pharmacology

Published: May 04, 2022

Hybrids of Imatinib with Quinoline: Synthesis, Antimyeloproliferative Activity Evaluation, and Molecular Docking.

Hybrids of Imatinib with Quinoline: Synthesis, Antimyeloproliferative Activity Evaluation, and Molecular Docking.

Journal: Pharmaceuticals (Basel, Switzerland)

Published: January 10, 2022

Comparative study between the anti-P. falciparum activity of triazolopyrimidine, pyrazolopyrimidine and quinoline derivatives and the identification of new PfDHODH inhibitors.

Comparative study between the anti-P. falciparum activity of triazolopyrimidine, pyrazolopyrimidine and quinoline derivatives and the identification of new PfDHODH inhibitors.

Journal: European journal of medicinal chemistry

Published: August 19, 2020

Synthesis of benzoylthiourea derivatives and analysis of their antibacterial performance against planktonic Staphylococcus aureus and its biofilms.

Synthesis of benzoylthiourea derivatives and analysis of their antibacterial performance against planktonic Staphylococcus aureus and its biofilms.

Journal: Letters in applied microbiology

Published: April 02, 2020

New pyrazolopyrimidine derivatives as Leishmania amazonensis arginase inhibitors.

New pyrazolopyrimidine derivatives as Leishmania amazonensis arginase inhibitors.

Journal: Bioorganic & medicinal chemistry

Published: March 22, 2019

Synthesis, Biological Evaluation, and Molecular Modeling Studies of New Thiadiazole Derivatives as Potent P2X7 Receptor Inhibitors.

Synthesis, Biological Evaluation, and Molecular Modeling Studies of New Thiadiazole Derivatives as Potent P2X7 Receptor Inhibitors.

Journal: Frontiers in chemistry

Published: January 21, 2019

New Efavirenz Derivatives and 1,2,3-Triazolyl-phosphonates as Inhibitors of Reverse Transcriptase of HIV-1.

New Efavirenz Derivatives and 1,2,3-Triazolyl-phosphonates as Inhibitors of Reverse Transcriptase of HIV-1.

Journal: Current topics in medicinal chemistry

Published: July 11, 2018

Evaluation of 7-arylaminopyrazolo[1,5-a]pyrimidines as anti-Plasmodium falciparum, antimalarial, and Pf-dihydroorotate dehydrogenase inhibitors.

Evaluation of 7-arylaminopyrazolo[1,5-a]pyrimidines as anti-Plasmodium falciparum, antimalarial, and Pf-dihydroorotate dehydrogenase inhibitors.

Journal: European journal of medicinal chemistry

Published: August 03, 2016

Synthesis, biological evaluation and molecular modeling of pseudo-peptides based statine as inhibitors for human tissue kallikrein 5.

Synthesis, biological evaluation and molecular modeling of pseudo-peptides based statine as inhibitors for human tissue kallikrein 5.

Journal: European journal of medicinal chemistry

Published: October 14, 2015

Molecular dynamics simulations of the free and inhibitor-bound cruzain systems in aqueous solvent: insights on the inhibition mechanism in acidic pH.

Molecular dynamics simulations of the free and inhibitor-bound cruzain systems in aqueous solvent: insights on the inhibition mechanism in acidic pH.

Journal: Journal of biomolecular structure & dynamics

Published: September 29, 2015

Structural and functional analysis of a platelet-activating lysophosphatidylcholine of Trypanosoma cruzi.

Structural and functional analysis of a platelet-activating lysophosphatidylcholine of Trypanosoma cruzi.

Journal: PLoS neglected tropical diseases

Published: December 18, 2013

Showing 1-12 of 13

Last Updated: 09/26/2026