Luiz A. Basso
Rio Grande, RS, Brazil
Last Updated: 09/26/2026
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Found 92 publications
Identification of Potential Anti-TB Candidates: A Step-by-Step Guide to Synthesis, MIC Determination, and Cytotoxicity Assessment in Mammalian Cells.
Journal: Journal of visualized experiments : JoVE
Published: June 08, 2026
4‑Aminoalkylquinolines as Potent Antitubercular Agents Targeting the Cytochrome bc1 Complex.
Journal: ACS medicinal chemistry letters
Published: April 06, 2026
Inhibitory effects of thiophene-2-thiazole hybrids against sensitive strains and resistant clinical isolates of Mycobacterium tuberculosis.
Journal: Bioorganic & medicinal chemistry letters
Published: March 06, 2026
Compartment-specific activation of kinin B1 and B2 receptors drives the production of vasoactive and inflammatory mediators during SARS-CoV-2 infection.
Journal: Immunology letters
Published: July 01, 2025
Scaffold Hopping Strategy toward New 4‑Aminoquinazolines Active Against Extracellular and Intracellular.
Journal: ACS medicinal chemistry letters
Published: May 12, 2025
In Vitro and In Silico Evaluation of Isatin-Derived Spirooxindoles as Antituberculosis Drug Candidates.
Journal: Chemical biology & drug design
Published: March 14, 2025
Preclinical Evaluation of Selene-Ethylenelacticamides in Tuberculosis: Effects Against Active, Dormant, and Resistant Mycobacterium Tuberculosis and In Vitro Toxicity Investigation.
Journal: Microorganisms
Published: January 15, 2025
Unveiling the Antimycobacterial Potential of Novel 4-Alkoxyquinolines: Insights into Selectivity, Mechanism of Action, and In Vivo Exposure.
Journal: Journal of medicinal chemistry
Published: December 04, 2024
Crystal structure of dihydroneopterin aldolase from Mycobacterium tuberculosis associated with 8-mercaptoguanine, and development of novel S8-functionalized analogues as inhibitors: Synthesis, enzyme inhibition, in vitro toxicity and antitubercular activity.
Journal: Journal of enzyme inhibition and medicinal chemistry
Published: August 14, 2024
Losartan and enalapril maleate differently influence SARS-CoV-2-infected vero cells.
Journal: Scientific reports
Published: July 01, 2024
Identification of antimycobacterial 8-hydroxyquinoline derivatives as in vitro enzymatic inhibitors of Mycobacterium tuberculosis enoyl-acyl carrier protein reductase.
Journal: Bioorganic chemistry
Published: May 08, 2024
Exploring Scaffold Hopping for Novel 2-(Quinolin-4-yloxy)acetamides with Enhanced Antimycobacterial Activity.
Journal: ACS medicinal chemistry letters
Published: December 20, 2023
Last Updated: 09/26/2026