Marc-antoine Bazin
Nantes, 44000, France
Last Updated: 09/26/2026
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Found 13 publications
5,6,7,8-Tetrahydroimidazo[1,2-a]pyrazine-based thiosemicarbazones as anti-Trypanosoma cruzi agents.
Journal: Bioorganic & medicinal chemistry
Published: January 24, 2026
Pharmacophore-guided optimization of the hit compound CTN1122 in the design of promising imidazo[1,2-a]pyrazine derivatives targeting the casein kinase 1 for antileishmanial therapy.
Journal: RSC medicinal chemistry
Published: March 25, 2025
Investigating the C2 Modulation of the Imidazo[1,2-a]pyrazine-Based Hit Compound CTN1122: Synthesis, in vitro Antileishmanial Activity, Cytotoxicity and Casein Kinase 1 Inhibition.
Journal: ChemMedChem
Published: October 29, 2024
Dibenzofuran Derivatives Inspired from Cercosporamide as Dual Inhibitors of Pim and CLK1 Kinases.
Journal: Molecules (Basel, Switzerland)
Published: October 04, 2021
In vitro identification of imidazo[1,2-a]pyrazine-based antileishmanial agents and evaluation of L. major casein kinase 1 inhibition.
Journal: European journal of medicinal chemistry
Published: September 04, 2020
Biological Evaluation of Arylsemicarbazone Derivatives as Potential Anticancer Agents.
Journal: Pharmaceuticals (Basel, Switzerland)
Published: October 10, 2019
5-Nitro-Thiophene-Thiosemicarbazone Derivatives Present Antitumor Activity Mediated by Apoptosis and DNA Intercalation.
Journal: Current topics in medicinal chemistry
Published: December 15, 2018
Benzofuro[3,2-d]pyrimidines inspired from cercosporamide CaPkc1 inhibitor: Synthesis and evaluation of fluconazole susceptibility restoration.
Journal: Bioorganic & medicinal chemistry letters
Published: March 28, 2018
Novel 1,6-naphthyridin-2(1H)-ones as potential anticancer agents targeting Hsp90.
Journal: European journal of medicinal chemistry
Published: February 03, 2016
Discovery of Novel (Imidazo[1,2-a]pyrazin-6-yl)ureas as Antiproliferative Agents Targeting P53 in Non-small Cell Lung Cancer Cell Lines.
Journal: Anticancer research
Published: January 22, 2016
Synthesis, antileishmanial activity and cytotoxicity of 2,3-diaryl- and 2,3,8-trisubstituted imidazo[1,2-a]pyrazines.
Journal: European journal of medicinal chemistry
Published: July 22, 2015
Synthesis and antiproliferative activity of benzofuran-based analogs of cercosporamide against non-small cell lung cancer cell lines.
Journal: European journal of medicinal chemistry
Published: July 16, 2013
Last Updated: 09/26/2026