Marc Le Borgne

Lyon, France

Last Updated: 09/26/2026

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Found 54 publications

Targeting Human Protein Kinase CK2 by a Library of Indeno[1,2-b]Indoles: Contribution of Thermal Shift Assay to Pre-Screening and Co-Crystallization to Post-Screening.

Targeting Human Protein Kinase CK2 by a Library of Indeno[1,2-b]Indoles: Contribution of Thermal Shift Assay to Pre-Screening and Co-Crystallization to Post-Screening.

Journal: Archiv der Pharmazie

Published: March 04, 2026

Identification of an N-methylpyrazole derivative as a selective inhibitor of breast cancer resistance protein (BCRP/ABCG2).

Identification of an N-methylpyrazole derivative as a selective inhibitor of breast cancer resistance protein (BCRP/ABCG2).

Journal: Archives of biochemistry and biophysics

Published: December 11, 2025

Formulation and Evaluation of Alginate Microcapsules Containing an Uncompetitive Nanomolar Dimeric Indenoindole Inhibitor of the Human Breast Cancer Resistance Pump ABCG2 with Different Excipients.

Formulation and Evaluation of Alginate Microcapsules Containing an Uncompetitive Nanomolar Dimeric Indenoindole Inhibitor of the Human Breast Cancer Resistance Pump ABCG2 with Different Excipients.

Journal: Pharmaceutics

Published: November 14, 2025

Functionalized nitrogen- and chalcogen-containing heterocyclic compounds as aromatase inhibitors: Design, synthesis and biological evaluation.

Functionalized nitrogen- and chalcogen-containing heterocyclic compounds as aromatase inhibitors: Design, synthesis and biological evaluation.

Journal: European journal of medicinal chemistry

Published: July 23, 2025

Exploring the biological potential of the brominated indenoindole MC11 and its interaction with protein kinase CK2.

Exploring the biological potential of the brominated indenoindole MC11 and its interaction with protein kinase CK2.

Journal: Biological chemistry

Published: December 15, 2024

Design, synthesis, and structure-activity relationship studies of 6H-benzo[b]indeno[1,2-d]thiophen-6-one derivatives as DYRK1A/CLK1/CLK4/haspin inhibitors.

Design, synthesis, and structure-activity relationship studies of 6H-benzo[b]indeno[1,2-d]thiophen-6-one derivatives as DYRK1A/CLK1/CLK4/haspin inhibitors.

Journal: RSC medicinal chemistry

Published: July 13, 2024

Antibody-drug conjugates: prospects for the next generation.

Antibody-drug conjugates: prospects for the next generation.

Journal: Drug discovery today

Published: July 02, 2024

New 2,4-bis[(substituted-aminomethyl)phenyl]phenylquinazoline and 2,4-bis[(substituted-aminomethyl)phenyl]phenylquinoline Derivatives: Synthesis and Biological Evaluation as Novel Anticancer Agents by Targeting G-Quadruplex.

New 2,4-bis[(substituted-aminomethyl)phenyl]phenylquinazoline and 2,4-bis[(substituted-aminomethyl)phenyl]phenylquinoline Derivatives: Synthesis and Biological Evaluation as Novel Anticancer Agents by Targeting G-Quadruplex.

Journal: Pharmaceuticals (Basel, Switzerland)

Published: November 11, 2023

Formulation and Investigation of CK2 Inhibitor-Loaded Alginate Microbeads with Different Excipients.

Formulation and Investigation of CK2 Inhibitor-Loaded Alginate Microbeads with Different Excipients.

Journal: Pharmaceutics

Published: October 31, 2023

Inhibitors of ABCG2-mediated multidrug resistance: Lead generation through computer-aided drug design.

Inhibitors of ABCG2-mediated multidrug resistance: Lead generation through computer-aided drug design.

Journal: European journal of medicinal chemistry

Published: October 22, 2022

Toxicological Risks of the Cobalt-Chromium Alloys in Dentistry: A Systematic Review.

Toxicological Risks of the Cobalt-Chromium Alloys in Dentistry: A Systematic Review.

Journal: Materials (Basel, Switzerland)

Published: July 07, 2022

Tetanus Toxin Fragment C: Structure, Drug Discovery Research and Production.

Tetanus Toxin Fragment C: Structure, Drug Discovery Research and Production.

Journal: Pharmaceuticals (Basel, Switzerland)

Published: May 20, 2022

Showing 1-12 of 54

Last Updated: 09/26/2026