Marielle Auberval
102 Avenue Gaston Roussel
Romainville, 93230, France
Romainville, 93230, France
Last Updated: 09/26/2026
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Found 8 publications
Anti-inflammatory, but not osteoprotective, effect of the TRAF6/CD40 inhibitor 6877002 in rodent models of local and systemic osteolysis.
Journal: Biochemical pharmacology
Published: October 20, 2021
Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases.
Journal: Journal of medicinal chemistry
Published: September 28, 2021
The Medium-Chain Fatty Acid Receptor GPR84 Mediates Myeloid Cell Infiltration Promoting Steatohepatitis and Fibrosis.
Journal: Journal of clinical medicine
Published: March 08, 2020
Neutralization of IL-17C Reduces Skin Inflammation in Mouse Models of Psoriasis and Atopic Dermatitis.
Journal: The Journal of investigative dermatology
Published: September 14, 2017
Discovery of 2-[[2-Ethyl-6-[4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]piperazin-1-yl]-8-methylimidazo[1,2-a]pyridin-3-yl]methylamino]-4-(4-fluorophenyl)thiazole-5-carbonitrile (GLPG1690), a First-in-Class Autotaxin Inhibitor Undergoing Clinical Evaluation for the Treatment of Idiopathic Pulmonary Fibrosis.
Journal: Journal of medicinal chemistry
Published: April 18, 2017
Characterization of GLPG0492, a selective androgen receptor modulator, in a mouse model of hindlimb immobilization.
Journal: BMC musculoskeletal disorders
Published: February 26, 2014
New potent calcimimetics: II. Discovery of benzothiazole trisubstituted ureas.
Journal: Bioorganic & medicinal chemistry letters
Published: November 09, 2012
New potent calcimimetics: I. Discovery of a series of novel trisubstituted ureas.
Journal: Bioorganic & medicinal chemistry letters
Published: November 09, 2012
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Last Updated: 09/26/2026