Masashi Yamasaki
Fujisawa, 2510012, Japan
Last Updated: 09/26/2026
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Found 14 publications
Design and Synthesis of Conformationally Constrained RORγt Inverse Agonists.
Journal: ChemMedChem
Published: July 12, 2019
Pharmacological evaluation of TAK-828F, a novel orally available RORγt inverse agonist, on murine chronic experimental autoimmune encephalomyelitis model.
Journal: Journal of neuroimmunology
Published: May 29, 2019
Pharmacological effects of TAK-828F: an orally available RORγt inverse agonist, in mouse colitis model and human blood cells of inflammatory bowel disease.
Journal: Inflammation research : official journal of the European Histamine Research Society ... [et al.]
Published: January 10, 2019
Pharmacological Inhibition of Toll-Like Receptor-4 Signaling by TAK242 Prevents and Induces Regression of Experimental Organ Fibrosis.
Journal: Frontiers in immunology
Published: April 25, 2018
Discovery of [ cis-3-({(5 R)-5-[(7-Fluoro-1,1-dimethyl-2,3-dihydro-1 H-inden-5-yl)carbamoyl]-2-methoxy-7,8-dihydro-1,6-naphthyridin-6(5 H)-yl}carbonyl)cyclobutyl]acetic Acid (TAK-828F) as a Potent, Selective, and Orally Available Novel Retinoic Acid Receptor-Related Orphan Receptor γt Inverse Agonist.
Journal: Journal of medicinal chemistry
Published: March 07, 2018
MLN3126, an antagonist of the chemokine receptor CCR9, ameliorates inflammation in a T cell mediated mouse colitis model.
Journal: International immunopharmacology
Published: February 08, 2018
Pharmacological inhibitory profile of TAK-828F, a potent and selective orally available RORγt inverse agonist.
Journal: Biochemical pharmacology
Published: November 14, 2017
Discovery of orally efficacious RORγt inverse agonists, part 1: Identification of novel phenylglycinamides as lead scaffolds.
Journal: Bioorganic & medicinal chemistry
Published: October 11, 2017
Discovery of orally efficacious RORγt inverse agonists. Part 2: Design, synthesis, and biological evaluation of novel tetrahydroisoquinoline derivatives.
Journal: Bioorganic & medicinal chemistry
Published: October 11, 2017
Identification of novel quinazolinedione derivatives as RORγt inverse agonist.
Journal: Bioorganic & medicinal chemistry
Published: October 09, 2017
Precise material identification method based on a photon counting technique with correction of the beam hardening effect in X-ray spectra.
Journal: Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine
Published: September 28, 2016
Last Updated: 09/26/2026