Mathilde Coevoet

Lille, 59000, France

Last Updated: 09/26/2026

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Found 13 publications

Towards the design of ligands of the internal pocket TEADs C-terminal domain.

Towards the design of ligands of the internal pocket TEADs C-terminal domain.

Journal: European journal of medicinal chemistry

Published: September 13, 2024

Novel Quinazoline Derivatives as Highly Effective A2A Adenosine Receptor Antagonists.

Novel Quinazoline Derivatives as Highly Effective A2A Adenosine Receptor Antagonists.

Journal: Molecules (Basel, Switzerland)

Published: July 11, 2024

Discovery of Compounds That Selectively Repress the Amyloidogenic Processing of the Amyloid Precursor Protein: Design, Synthesis and Pharmacological Evaluation of Diphenylpyrazoles.

Discovery of Compounds That Selectively Repress the Amyloidogenic Processing of the Amyloid Precursor Protein: Design, Synthesis and Pharmacological Evaluation of Diphenylpyrazoles.

Journal: International journal of molecular sciences

Published: September 20, 2022

High ligand efficiency quinazoline compounds as novel A2A adenosine receptor antagonists.

High ligand efficiency quinazoline compounds as novel A2A adenosine receptor antagonists.

Journal: European journal of medicinal chemistry

Published: January 12, 2022

Discovery of a cryptic site at the interface 2 of TEAD - Towards a new family of YAP/TAZ-TEAD inhibitors.

Discovery of a cryptic site at the interface 2 of TEAD - Towards a new family of YAP/TAZ-TEAD inhibitors.

Journal: European journal of medicinal chemistry

Published: July 02, 2021

Design, Synthesis and Evaluation of a Series of 1,5-Diaryl-1,2,3-triazole-4-carbohydrazones as Inhibitors of the YAP-TAZ/TEAD Complex.

Design, Synthesis and Evaluation of a Series of 1,5-Diaryl-1,2,3-triazole-4-carbohydrazones as Inhibitors of the YAP-TAZ/TEAD Complex.

Journal: ChemMedChem

Published: March 03, 2021

New piperazine multi-effect drugs prevent neurofibrillary degeneration and amyloid deposition, and preserve memory in animal models of Alzheimer's disease.

New piperazine multi-effect drugs prevent neurofibrillary degeneration and amyloid deposition, and preserve memory in animal models of Alzheimer's disease.

Journal: Neurobiology of disease

Published: July 24, 2018

Contribution of the Endosomal-Lysosomal and Proteasomal Systems in Amyloid-β Precursor Protein Derived Fragments Processing.

Contribution of the Endosomal-Lysosomal and Proteasomal Systems in Amyloid-β Precursor Protein Derived Fragments Processing.

Journal: Frontiers in cellular neuroscience

Published: July 05, 2018

A phenotypic approach to the discovery of compounds that promote non-amyloidogenic processing of the amyloid precursor protein: Toward a new profile of indirect β-secretase inhibitors.

A phenotypic approach to the discovery of compounds that promote non-amyloidogenic processing of the amyloid precursor protein: Toward a new profile of indirect β-secretase inhibitors.

Journal: European journal of medicinal chemistry

Published: July 04, 2018

Toward the Discovery of a Novel Class of YAP⁻TEAD Interaction Inhibitors by Virtual Screening Approach Targeting YAP⁻TEAD Protein⁻Protein Interface.

Toward the Discovery of a Novel Class of YAP⁻TEAD Interaction Inhibitors by Virtual Screening Approach Targeting YAP⁻TEAD Protein⁻Protein Interface.

Journal: Cancers

Published: April 24, 2018

Design and synthesis of 2,6-disubstituted-8-amino imidazo[1,2a]pyridines, a promising privileged structure.

Design and synthesis of 2,6-disubstituted-8-amino imidazo[1,2a]pyridines, a promising privileged structure.

Journal: Bioorganic & medicinal chemistry

Published: March 09, 2018

New phenylaniline derivatives as modulators of amyloid protein precursor metabolism.

New phenylaniline derivatives as modulators of amyloid protein precursor metabolism.

Journal: Bioorganic & medicinal chemistry

Published: December 22, 2017

Showing 1-12 of 13

Last Updated: 09/26/2026