Maurizio Anzini
Via Aldo Moro 2
Siena, 53100, Italy
Siena, 53100, Italy
Last Updated: 09/26/2026
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Found 36 publications
Evaluation of a New Riluzole-Based Compound VA945 on Sodium and Potassium Conductances Expressed by SH-SY5Y- Derived Neurons.
Journal: Journal of neurochemistry
Published: July 24, 2025
VA1213, a selective COX-2 inhibitor, exhibits antitumor activity by suppressing EGFR, AKT, and ERK1/2 phosphorylation.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences
Published: July 22, 2025
Use of imidazo[1,5-a]quinoline scaffold as the pharmacophore in the design of bivalent ligands of central benzodiazepine receptors.
Journal: Bioorganic & medicinal chemistry
Published: August 13, 2024
Novel multitarget directed ligands inspired by riluzole: A serendipitous synthesis of substituted benzo[b][1,4]thiazepines potentially useful as neuroprotective agents.
Journal: Bioorganic & medicinal chemistry
Published: July 22, 2024
Novel analgesic/anti-inflammatory agents: 1,5-Diarylpyrrole nitrooxyethyl sulfides and related compounds as Cyclooxygenase-2 inhibitors containing a nitric oxide donor moiety endowed with vasorelaxant properties.
Journal: European journal of medicinal chemistry
Published: May 04, 2022
Exploring Translocator Protein (TSPO) Medicinal Chemistry: An Approach for Targeting Radionuclides and Boron Atoms to Mitochondria.
Journal: Journal of medicinal chemistry
Published: July 13, 2021
Therapeutic potential for coxibs-nitric oxide releasing hybrids in cystic fibrosis.
Journal: European journal of medicinal chemistry
Published: June 04, 2020
Design, synthesis and biological evaluation of 7-substituted 4-phenyl-6H-imidazo[1,5-a]thieno[3,2-f] [1,4]diazepines as safe anxiolytic agents.
Journal: European journal of medicinal chemistry
Published: February 25, 2020
Synthesis, biological evaluation and molecular modeling of novel selective COX-2 inhibitors: sulfide, sulfoxide, and sulfone derivatives of 1,5-diarylpyrrol-3-substituted scaffold.
Journal: Bioorganic & medicinal chemistry
Published: June 27, 2019
Radiosynthesis and Preclinical Evaluation of 11C-VA426, a Cyclooxygenase-2 Selective Ligand.
Journal: Contrast media & molecular imaging
Published: March 01, 2019
Last Updated: 09/26/2026