Mauro Niso
Bari, Italy
Last Updated: 09/26/2026
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Found 64 publications
A Novel Class of "Super-Strained" Spiro Heterocycles: Gateway to 1-Azaspiro[3.3]heptane Derivatives, and Biological Validation.
Journal: Angewandte Chemie (International ed. in English)
Published: March 24, 2026
Development of Second-Generation Phenoxyethylpiperidines as Potent Sigma-1 Receptor Agonists with Neuroprotective Potential for Alzheimer's Disease.
Journal: Journal of medicinal chemistry
Published: February 05, 2026
Correction to "First-In-Class Thiosemicarbazone Metal Complexes Targeting the Sigma-2 Receptor (S2R) as an Innovative Strategy against Pancreatic Cancer".
Journal: Journal of medicinal chemistry
Published: January 16, 2026
A Holistic Approach to Identifying a Positron Emission Tomography (PET) Tracer Candidate for In Vivo Imaging of Purinergic P2X7 Receptor in Neuroinflammation.
Journal: ACS pharmacology & translational science
Published: December 23, 2025
Development of dual acting selenium-doped hydroxyapatite nanoparticles with platinum-bisphosphonate complexes for bone cancer therapy.
Journal: RSC advances
Published: December 03, 2025
Hydrogen Sulfide (H2S)-Donating Formyl Peptide Receptor 2 (FPR2) Agonists: Design, Synthesis, and Biological Evaluation in Primary Mouse Microglia Culture.
Journal: Antioxidants (Basel, Switzerland)
Published: June 04, 2025
New oxaliplatin-zoledronate derivatives with potential antitumor activity towards bone tumors and metastases.
Journal: Journal of inorganic biochemistry
Published: February 07, 2025
Exploring Selenium-Functionalized Hydroxyapatite Using Organic Selenocystine for Antitumor Applications.
Journal: Materials (Basel, Switzerland)
Published: January 30, 2025
First-In-Class Thiosemicarbazone Metal Complexes Targeting the Sigma-2 Receptor (S2R) as an Innovative Strategy against Pancreatic Cancer.
Journal: Journal of medicinal chemistry
Published: November 18, 2024
Nature-Inspired 1-Phenylpyrrolo[2,1-a]isoquinoline Scaffold for Novel Antiproliferative Agents Circumventing P-Glycoprotein-Dependent Multidrug Resistance.
Journal: Pharmaceuticals (Basel, Switzerland)
Published: March 06, 2024
In-vitro and in-silico studies of annelated 1,4,7,8-tetrahydroazocine ester derivatives as nanomolar selective inhibitors of human butyrylcholinesterase.
Journal: Chemico-biological interactions
Published: August 04, 2023
Cytotoxic pathways activated by multifunctional thiosemicarbazones targeting sigma-2 receptors in breast and lung carcinoma cells.
Journal: Pharmacological reports : PR
Published: June 22, 2023
Last Updated: 09/26/2026