Mona F. Said
Kasr El Aini Street
Cairo, C 11562, Egypt
Cairo, C 11562, Egypt
Last Updated: 09/26/2026
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Found 25 publications
Design and discovery of 1,4-dihydropyrimidinone-based noncovalent DprE1 inhibitors with integrated biological and computational validation against Mycobacterium tuberculosis.
Journal: Bioorganic chemistry
Published: May 26, 2026
In vitro, in vivo, and in silico profiling of optimized hydrazide-hydrazone indole congeners as multi-faceted AChE, BACE1, and MAO-B inhibitors for Alzheimer's disease therapy.
Journal: Bioorganic chemistry
Published: January 17, 2026
Targeting EGFR With Quinazoline-4-One/Chalcone Hybrids: Design, Synthesis, and Anticancer Evaluation.
Journal: Archiv der Pharmazie
Published: September 27, 2025
Design and synthesis of novel 3,5-diphenyl pyrazolines acting as potent EGFR inhibitors with off-target antileukemic effect.
Journal: Future medicinal chemistry
Published: September 15, 2025
Probing new 3-hydrazinyl indole phenacetamide derivatives as multitarget anti-Alzheimer: Synthesis, in vivo, in vitro, and in silico studies.
Journal: European journal of medicinal chemistry
Published: March 18, 2025
3,5-Disubstituted pyrazoline as a promising core for anticancer agents: mechanisms of action and therapeutic potentials.
Journal: Future medicinal chemistry
Published: March 13, 2025
Novel isatin conjugates endowed with analgesic and anti-inflammatory properties: design, synthesis and biological evaluation.
Journal: Future medicinal chemistry
Published: December 16, 2024
6,7-Dimethoxy-2-methyl-4-substituted quinazolines: Design, synthesis, EGFR inhibitory activity, in vitro cytotoxicity, and in silico studies.
Journal: European journal of medicinal chemistry
Published: November 12, 2024
Insight on novel sulfamoylphenyl pyrazole derivatives as anticancer carbonic anhydrase inhibitors.
Journal: Molecular diversity
Published: September 01, 2024
Exploring of novel oxazolones and imidazolones as anti-inflammatory and analgesic candidates with cyclooxygenase inhibitory action.
Journal: Future medicinal chemistry
Published: April 19, 2024
Insight on novel oxindole conjugates adopting different anti-inflammatory investigations and quantitative evaluation.
Journal: Future medicinal chemistry
Published: April 18, 2024
Exploring new imines as anti-inflammatory COX and 5-LOX inhibitors with an improved pharmacokinetic profile.
Journal: Future medicinal chemistry
Published: January 31, 2024
Last Updated: 09/26/2026