Nizar A. Al-Shar'i
Irbid, IR, Jordan
Last Updated: 09/26/2026
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Found 37 publications
PTUPB, a soluble epoxide hydrolase/cyclooxygenase‑2 dual inhibitor, reduces endothelial‑to‑mesenchymal transition and improves doxorubicin‑induced vascular and cardiac toxicity.
Journal: Molecular medicine reports
Published: March 18, 2025
Anticancer and Cyclooxygenase Inhibitory Activity of Benzylidene Derivatives of Fenobam and its Thio Analogues.
Journal: Current medicinal chemistry
Published: August 16, 2024
Anticancer and Cyclooxygenase Inhibitory Activity of Benzylidene Derivatives of Fenobam and its Thio Analogues.
Journal: Current medicinal chemistry
Published: August 16, 2024
The design of TOPK inhibitors using similarity search, molecular docking, and MD simulations.
Journal: Journal of biomolecular structure & dynamics
Published: February 15, 2024
Synthesis, characterization and larvicidal studies of ethyl 3-benzoyl-7-(piperidin-1-yl)indolizine-1-carboxylate analogues against Anopheles arabiensis and cheminformatics approaches.
Journal: Journal of biomolecular structure & dynamics
Published: February 05, 2024
Identification of potent indolizine derivatives against Mycobacterial tuberculosis: In vitro anti-TB properties, in silico target validation, molecular docking and dynamics studies.
Journal: International journal of biological macromolecules
Published: November 20, 2023
Synthesis, biological evaluation, and computational investigation of ethyl 2,4,6-trisubstituted-1,4-dihydropyrimidine-5-carboxylates as potential larvicidal agents against Anopheles arabiensis.
Journal: Journal of biomolecular structure & dynamics
Published: June 01, 2023
Antitubercular, Cytotoxicity, and Computational Target Validation of Dihydroquinazolinone Derivatives.
Journal: Antibiotics (Basel, Switzerland)
Published: May 30, 2022
Evaluation of EDTA Dianhydride Versus Diphenyl Carbonate Nanosponges for Curcumin.
Journal: AAPS PharmSciTech
Published: May 01, 2022
The impact of cycleanine in cancer research: a computational study.
Journal: Journal of molecular modeling
Published: April 08, 2022
1,2,3-Triazolyl-tetrahydropyrimidine Conjugates as Potential Sterol Carrier Protein-2 Inhibitors: Larvicidal Activity against the Malaria Vector Anopheles arabiensis and In Silico Molecular Docking Study.
Journal: Molecules (Basel, Switzerland)
Published: March 05, 2022
Weak complexation of 5-fluorouracil with β-cyclodextrin, carbonate, and dianhydride crosslinked β-cyclodextrin: in vitro and in silico studies.
Journal: Research in pharmaceutical sciences
Published: December 16, 2021
Last Updated: 09/26/2026