Pravin S. Iyer
Bellary Road, Hebbal
Bengaluru, KA 560024, India
Bengaluru, KA 560024, India
Last Updated: 09/26/2026
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Found 19 publications
Discovery of aminopiperidine based potent & novel topoisomerase inhibitor with broad spectrum anti-bacterial activity.
Journal: Bioorganic & medicinal chemistry letters
Published: March 26, 2024
Discovery of N-Cyano-sulfoximineurea Derivatives as Potent and Orally Bioavailable NLRP3 Inflammasome Inhibitors.
Journal: ACS medicinal chemistry letters
Published: September 19, 2019
Scaffold Morphing To Identify Novel DprE1 Inhibitors with Antimycobacterial Activity.
Journal: ACS medicinal chemistry letters
Published: July 29, 2019
Design and synthesis of functionalized piperazin-1yl-(E)-stilbenes as inhibitors of 17α-hydroxylase-C17,20-lyase (Cyp17).
Journal: Bioorganic & medicinal chemistry letters
Published: January 30, 2018
Discovery of Imidazo[1,2-a]pyridine Ethers and Squaramides as Selective and Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthesis.
Journal: Journal of medicinal chemistry
Published: January 12, 2017
Design, synthesis, and evaluation of (2S,4R)-Ketoconazole sulfonamide analogs as potential treatments for Metabolic Syndrome.
Journal: Bioorganic & medicinal chemistry letters
Published: June 25, 2016
Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate.
Journal: Nature communications
Published: September 15, 2014
Synthesis and in vitro evaluation of novel 8-aminoquinoline-pyrazolopyrimidine hybrids as potent antimalarial agents.
Journal: Bioorganic & medicinal chemistry letters
Published: August 13, 2014
Synthesis and biological evaluation of adamantane-based aminophenols as a novel class of antiplasmodial agents.
Journal: Bioorganic & medicinal chemistry letters
Published: August 13, 2014
N-aryl-2-aminobenzimidazoles: novel, efficacious, antimalarial lead compounds.
Journal: Journal of medicinal chemistry
Published: July 10, 2014
1,4-azaindole, a potential drug candidate for treatment of tuberculosis.
Journal: Antimicrobial agents and chemotherapy
Published: June 25, 2014
Aminoazabenzimidazoles, a novel class of orally active antimalarial agents.
Journal: Journal of medicinal chemistry
Published: June 11, 2014
Last Updated: 09/26/2026