Rafael Castillo
Ciudad De México C.P. 04510
Mexico, MEX 04510, Mexico
Mexico, MEX 04510, Mexico
Last Updated: 09/26/2026
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Found 56 publications
Fosfatriclaben: Effective dose determination and comparative efficacy assessment with closantel, triclabendazole+ivermectin, triclabendazole+albendazole in artificially infected cattle.
Journal: Experimental parasitology
Published: May 19, 2024
Inhibition of Shikimate Kinase from Methicillin-Resistant Staphylococcus aureus by Benzimidazole Derivatives. Kinetic, Computational, Toxicological, and Biological Activity Studies.
Journal: International journal of molecular sciences
Published: March 15, 2024
Influence of extracellular ATP on mammalian sperm physiology.
Journal: Reproduction, fertility, and development
Published: December 14, 2023
Characterization of the Effect of N-(2-Methoxyphenyl)-1-methyl-1H-benzimidazol-2-amine, Compound 8, against Leishmania mexicana and Its In Vivo Leishmanicidal Activity.
Journal: International journal of molecular sciences
Published: December 01, 2023
Structure-Based Optimization of Carbendazim-Derived Tubulin Polymerization Inhibitors through Alchemical Free Energy Calculations.
Journal: Journal of chemical information and modeling
Published: November 10, 2023
Fosfatriclaben, a prodrug of triclabendazole: Preparation, stability, and fasciolicidal activity of three new intramuscular formulations.
Journal: Veterinary parasitology
Published: August 25, 2023
Development and Pharmacokinetic Evaluation of Two Parenteral Formulations of Albendazole Using Prodrug and Cosolvent Approaches.
Journal: AAPS PharmSciTech
Published: April 14, 2023
Garbage in, garbage out: how reliable training data improved a virtual screening approach against SARS-CoV-2 MPro.
Journal: Frontiers in pharmacology
Published: March 24, 2023
Computational Methods in Cooperation with Experimental Approaches to Design Protein Tyrosine Phosphatase 1B Inhibitors in Type 2 Diabetes Drug Design: A Review of the Achievements of This Century.
Journal: Pharmaceuticals (Basel, Switzerland)
Published: June 11, 2022
Structure-Activity Relationship of N-Phenylthieno[2,3-b]pyridine-2-carboxamide Derivatives Designed as Forkhead Box M1 Inhibitors: The Effect of Electron-Withdrawing and Donating Substituents on the Phenyl Ring.
Journal: Pharmaceuticals (Basel, Switzerland)
Published: January 16, 2022
Benzimidazole Derivatives as New and Selective Inhibitors of Arginase from Leishmania mexicana with Biological Activity against Promastigotes and Amastigotes.
Journal: International journal of molecular sciences
Published: December 01, 2021
Design, synthesis, kinetic, molecular dynamics, and hypoglycemic effect characterization of new and potential selective benzimidazole derivatives as Protein Tyrosine Phosphatase 1B inhibitors.
Journal: Bioorganic & medicinal chemistry
Published: July 08, 2021
Last Updated: 09/26/2026