Last Updated: 09/26/2026
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Found 2 publications
Optimization of α-Fluoro, β-Heteroaryl Acrylamide Warheads for KRASG12C Active-State Inhibition.
Journal: Journal of medicinal chemistry
Published: March 02, 2026
Covalent inhibitor design confers activity against both GDP- and GTP-bound forms of KRAS G12C.
Journal: Nature communications
Published: March 03, 2025
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Last Updated: 09/26/2026