Robert Foltyn-Frank

Aachen, NW 52078, Germany

Last Updated: 09/26/2026

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Found 14 publications

2-(Halogenated Phenyl) acetamides and propanamides as potent TRPV1 antagonists.

2-(Halogenated Phenyl) acetamides and propanamides as potent TRPV1 antagonists.

Journal: Bioorganic & medicinal chemistry letters

Published: June 14, 2021

Discovery of 1-(1H-indazol-4-yl)-3-((1-phenyl-1H-pyrazol-5-yl)methyl) ureas as potent and thermoneutral TRPV1 antagonists.

Discovery of 1-(1H-indazol-4-yl)-3-((1-phenyl-1H-pyrazol-5-yl)methyl) ureas as potent and thermoneutral TRPV1 antagonists.

Journal: Bioorganic & medicinal chemistry letters

Published: July 21, 2020

Discovery of indane propanamides as potent and selective TRPV1 antagonists.

Discovery of indane propanamides as potent and selective TRPV1 antagonists.

Journal: Bioorganic & medicinal chemistry letters

Published: October 17, 2019

In vitro characterization of the thermoneutral transient receptor potential vanilloid-1 (TRPV1) inhibitor GRTE16523.

In vitro characterization of the thermoneutral transient receptor potential vanilloid-1 (TRPV1) inhibitor GRTE16523.

Journal: European journal of pharmacology

Published: July 30, 2019

4-Aminophenyl acetamides and propanamides as potent transient receptor potential vanilloid 1 (TRPV1) ligands.

4-Aminophenyl acetamides and propanamides as potent transient receptor potential vanilloid 1 (TRPV1) ligands.

Journal: Bioorganic & medicinal chemistry

Published: July 09, 2018

Discovery of 2-(3,5-difluoro-4-methylsulfonaminophenyl)propanamides as potent TRPV1 antagonists.

Discovery of 2-(3,5-difluoro-4-methylsulfonaminophenyl)propanamides as potent TRPV1 antagonists.

Journal: Bioorganic & medicinal chemistry letters

Published: March 19, 2018

Pyrazole C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

Pyrazole C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

Journal: Bioorganic & medicinal chemistry letters

Published: July 04, 2017

t-Butyl pyridine and phenyl C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

t-Butyl pyridine and phenyl C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

Journal: Bioorganic & medicinal chemistry

Published: February 14, 2017

Structure activity relationships of benzyl C-region analogs of 2-(3-fluoro-4-methylsulfonamidophenyl)propanamides as potent TRPV1 antagonists.

Structure activity relationships of benzyl C-region analogs of 2-(3-fluoro-4-methylsulfonamidophenyl)propanamides as potent TRPV1 antagonists.

Journal: Bioorganic & medicinal chemistry

Published: September 05, 2015

α-Substituted 2-(3-fluoro-4-methylsulfonamidophenyl)acetamides as potent TRPV1 antagonists.

α-Substituted 2-(3-fluoro-4-methylsulfonamidophenyl)acetamides as potent TRPV1 antagonists.

Journal: Bioorganic & medicinal chemistry letters

Published: March 06, 2015

Pyridine C-region analogs of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

Pyridine C-region analogs of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

Journal: European journal of medicinal chemistry

Published: December 03, 2014

6,6-Fused heterocyclic ureas as highly potent TRPV1 antagonists.

6,6-Fused heterocyclic ureas as highly potent TRPV1 antagonists.

Journal: Bioorganic & medicinal chemistry letters

Published: December 03, 2014

Showing 1-12 of 14

Last Updated: 09/26/2026