Roland Blanque
Romainville, France
Last Updated: 09/26/2026
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Found 12 publications
Pharmacological Characterization of GLPG3667, a Tyrosine Kinase 2-Selective Inhibitor, for the Treatment of Inflammatory and Autoimmune Diseases.
Journal: Inflammation
Published: December 24, 2025
Discovery of GLPG4471, a potent and selective IRAK4 inhibitor for the treatment of inflammatory and autoimmune diseases.
Journal: Bioorganic & medicinal chemistry letters
Published: June 27, 2025
GLPG2737, a CFTR Inhibitor, Prevents Cyst Growth in Preclinical Models of Autosomal Dominant Polycystic Kidney Disease.
Journal: American journal of nephrology
Published: August 29, 2024
Discovery of GLPG3667, a Selective ATP Competitive Tyrosine Kinase 2 Inhibitor for the Treatment of Autoimmune Diseases.
Journal: Journal of medicinal chemistry
Published: May 28, 2024
Pharmacological characterization of GLPG1972/S201086, a potent and selective small-molecule inhibitor of ADAMTS5.
Journal: Osteoarthritis and cartilage
Published: March 15, 2021
Discovery of GLPG1972/S201086, a Potent, Selective, and Orally Bioavailable ADAMTS-5 Inhibitor for the Treatment of Osteoarthritis.
Journal: Journal of medicinal chemistry
Published: March 15, 2021
Discovery of 9-Cyclopropylethynyl-2-((S)-1-[1,4]dioxan-2-ylmethoxy)-6,7-dihydropyrimido[6,1-a]isoquinolin-4-one (GLPG1205), a Unique GPR84 Negative Allosteric Modulator Undergoing Evaluation in a Phase II Clinical Trial.
Journal: Journal of medicinal chemistry
Published: September 09, 2020
Population Pharmacokinetic and Pharmacodynamic Analysis of GLPG1690, an Autotaxin Inhibitor, in Healthy Volunteers and Patients with Idiopathic Pulmonary Fibrosis.
Journal: Clinical pharmacokinetics
Published: April 07, 2019
Discovery of 2-[[2-Ethyl-6-[4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]piperazin-1-yl]-8-methylimidazo[1,2-a]pyridin-3-yl]methylamino]-4-(4-fluorophenyl)thiazole-5-carbonitrile (GLPG1690), a First-in-Class Autotaxin Inhibitor Undergoing Clinical Evaluation for the Treatment of Idiopathic Pulmonary Fibrosis.
Journal: Journal of medicinal chemistry
Published: April 18, 2017
Discovery and optimization of an azetidine chemical series as a free fatty acid receptor 2 (FFA2) antagonist: from hit to clinic.
Journal: Journal of medicinal chemistry
Published: November 08, 2014
Characterization of GLPG0492, a selective androgen receptor modulator, in a mouse model of hindlimb immobilization.
Journal: BMC musculoskeletal disorders
Published: February 26, 2014
Identification of a 4-(hydroxymethyl)diarylhydantoin as a selective androgen receptor modulator.
Journal: Journal of medicinal chemistry
Published: September 11, 2012
Showing 1-12 of 12
Last Updated: 09/26/2026