Santiago B. Ferrer
Tres Cantos, MD, Spain
Last Updated: 09/26/2026
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Found 27 publications
Prediction of lung exposure to anti-tubercular drugs using plasma pharmacokinetic data: Implications for dose selection.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences
Published: June 27, 2021
Design and tests of prospective property predictions for novel antimalarial 2-aminopropylaminoquinolones.
Journal: Journal of computer-aided molecular design
Published: April 09, 2020
Lead Optimization of a Pyrrole-Based Dihydroorotate Dehydrogenase Inhibitor Series for the Treatment of Malaria.
Journal: Journal of medicinal chemistry
Published: April 07, 2020
Identification of GSK3186899/DDD853651 as a Preclinical Development Candidate for the Treatment of Visceral Leishmaniasis.
Journal: Journal of medicinal chemistry
Published: December 21, 2018
Identification of Fast-Acting 2,6-Disubstituted Imidazopyridines That Are Efficacious in the in Vivo Humanized Plasmodium falciparum NODscidIL2Rγ null Mouse Model of Malaria.
Journal: Journal of medicinal chemistry
Published: April 19, 2018
Synthesis and Structure-Activity Relationships of the Novel Antimalarials 5-Pyridinyl-4(1 H)-Pyridones.
Journal: Journal of medicinal chemistry
Published: March 29, 2018
A human microdose study of the antimalarial drug GSK3191607 in healthy volunteers.
Journal: British journal of clinical pharmacology
Published: August 11, 2017
A potent series targeting the malarial cGMP-dependent protein kinase clears infection and blocks transmission.
Journal: Nature communications
Published: February 20, 2017
Identification of a Potential Antimalarial Drug Candidate from a Series of 2-Aminopyrazines by Optimization of Aqueous Solubility and Potency across the Parasite Life Cycle.
Journal: Journal of medicinal chemistry
Published: October 18, 2016
The multistate tuberculosis pharmacometric model: a semi-mechanistic pharmacokinetic-pharmacodynamic model for studying drug effects in an acute tuberculosis mouse model.
Journal: Journal of pharmacokinetics and pharmacodynamics
Published: September 08, 2016
Trisubstituted Pyrimidines as Efficacious and Fast-Acting Antimalarials.
Journal: Journal of medicinal chemistry
Published: June 18, 2016
Population pharmacokinetics, optimised design and sample size determination for rifampicin, isoniazid, ethambutol and pyrazinamide in the mouse.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences
Published: February 22, 2016
Last Updated: 09/26/2026