Last Updated: 09/26/2026
Save publications for later
Sign Up
Not sure about your diagnosis?
Check Your Symptoms
Found 6 publications
Discovery of [11C]MK-6884: A Positron Emission Tomography (PET) Imaging Agent for the Study of M4Muscarinic Receptor Positive Allosteric Modulators (PAMs) in Neurodegenerative Diseases.
Journal: Journal of medicinal chemistry
Published: February 27, 2020
Discovery, Optimization, and Biological Characterization of 2,3,6-Trisubstituted Pyridine-Containing M4 Positive Allosteric Modulators.
Journal: ChemMedChem
Published: February 11, 2019
Extending 'predict first' to the design-make-test cycle in small-molecule drug discovery.
Journal: Future medicinal chemistry
Published: April 14, 2017
Synthesis and optimization of N-heterocyclic pyridinones as catechol-O-methyltransferase (COMT) inhibitors.
Journal: Bioorganic & medicinal chemistry letters
Published: February 09, 2016
Synthesis and Evaluation of Heterocyclic Catechol Mimics as Inhibitors of Catechol-O-methyltransferase (COMT).
Journal: ACS medicinal chemistry letters
Published: December 05, 2014
Characterization of non-nitrocatechol pan and isoform specific catechol-O-methyltransferase inhibitors and substrates.
Journal: ACS chemical neuroscience
Published: November 01, 2011
Showing 1-6 of 6
Last Updated: 09/26/2026