Simon F. Campbell
ICC, Route De Pré Bois 20
Geneve, GE 1215, Switzerland
Geneve, GE 1215, Switzerland
Last Updated: 09/26/2026
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Found 15 publications
Optimization of Species-Selective Reversible Proteasome Inhibitors for the Treatment of Malaria.
Journal: Journal of medicinal chemistry
Published: October 28, 2025
Identification of potent and reversible piperidine carboxamides that are species-selective orally active proteasome inhibitors to treat malaria.
Journal: Cell chemical biology
Published: March 04, 2024
Hit-to-lead optimization of a 2-aminobenzimidazole series as new candidates for chagas disease.
Journal: European journal of medicinal chemistry
Published: September 25, 2022
Discovery and Preclinical Pharmacology of INE963, a Potent and Fast-Acting Blood-Stage Antimalarial with a High Barrier to Resistance and Potential for Single-Dose Cures in Uncomplicated Malaria.
Journal: Journal of medicinal chemistry
Published: March 01, 2022
Hit-to-lead optimization of a benzene sulfonamide series for potential antileishmanial agents.
Journal: RSC medicinal chemistry
Published: June 04, 2021
The antimalarial MMV688533 provides potential for single-dose cures with a high barrier to Plasmodium falciparum parasite resistance.
Journal: Science translational medicine
Published: January 15, 2021
2-aminobenzimidazoles for leishmaniasis: From initial hit discovery to in vivo profiling.
Journal: PLoS neglected tropical diseases
Published: September 10, 2020
Substituted Aminoacetamides as Novel Leads for Malaria Treatment.
Journal: ChemMedChem
Published: June 01, 2019
2,3,8-Trisubstituted Quinolines with Antimalarial Activity.
Journal: Anais da Academia Brasileira de Ciencias
Published: October 13, 2017
Novel inhibitors of Plasmodium falciparum based on 2,5-disubstituted furans.
Journal: European journal of medicinal chemistry
Published: October 31, 2016
Discovery of a Quinoline-4-carboxamide Derivative with a Novel Mechanism of Action, Multistage Antimalarial Activity, and Potent in Vivo Efficacy.
Journal: Journal of medicinal chemistry
Published: September 16, 2016
A tetraoxane-based antimalarial drug candidate that overcomes PfK13-C580Y dependent artemisinin resistance.
Journal: Nature communications
Published: September 02, 2016
Last Updated: 09/26/2026