Simon F. Macdonald

Stevenage, ENG SG12NY, United Kingdom

Last Updated: 09/26/2026

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Found 51 publications

Core Modifications of GSK3335103 toward Orally Bioavailable αvβ6 Inhibitors with Improved Synthetic Tractability.

Core Modifications of GSK3335103 toward Orally Bioavailable αvβ6 Inhibitors with Improved Synthetic Tractability.

Journal: Journal of medicinal chemistry

Published: October 17, 2024

Discovery and Development of Highly Potent and Orally Bioavailable Nonpeptidic αvβ6 Integrin Inhibitors.

Discovery and Development of Highly Potent and Orally Bioavailable Nonpeptidic αvβ6 Integrin Inhibitors.

Journal: Journal of medicinal chemistry

Published: September 13, 2024

Structure-Based Design of a Novel Class of Autotaxin Inhibitors Based on Endogenous Allosteric Modulators.

Structure-Based Design of a Novel Class of Autotaxin Inhibitors Based on Endogenous Allosteric Modulators.

Journal: Journal of medicinal chemistry

Published: April 20, 2022

How Diverse Is Medicinal Chemistry? Insights into Race, Ethnicity, Origin, Gender, and Geography.

How Diverse Is Medicinal Chemistry? Insights into Race, Ethnicity, Origin, Gender, and Geography.

Journal: Journal of medicinal chemistry

Published: December 21, 2021

Pharmacological characterisation of GSK3335103, an oral αvβ6 integrin small molecule RGD-mimetic inhibitor for the treatment of fibrotic disease.

Pharmacological characterisation of GSK3335103, an oral αvβ6 integrin small molecule RGD-mimetic inhibitor for the treatment of fibrotic disease.

Journal: European journal of pharmacology

Published: September 30, 2021

Emerging therapeutic opportunities for integrin inhibitors.

Emerging therapeutic opportunities for integrin inhibitors.

Journal: Nature reviews. Drug discovery

Published: July 26, 2021

Writing Your Next Medicinal Chemistry Article: Journal Bibliometrics and Guiding Principles for Industrial Authors.

Writing Your Next Medicinal Chemistry Article: Journal Bibliometrics and Guiding Principles for Industrial Authors.

Journal: Journal of medicinal chemistry

Published: October 26, 2020

Iridium-catalysed C-H borylation of β-aryl-aminopropionic acids.

Iridium-catalysed C-H borylation of β-aryl-aminopropionic acids.

Journal: Organic & biomolecular chemistry

Published: September 02, 2020

Correction to: Heparin resistance in COVID‑19 patients in the intensive care unit.

Correction to: Heparin resistance in COVID‑19 patients in the intensive care unit.

Journal: Journal of thrombosis and thrombolysis

Published: June 24, 2020

Heparin resistance in COVID-19 patients in the intensive care unit.

Heparin resistance in COVID-19 patients in the intensive care unit.

Journal: Journal of thrombosis and thrombolysis

Published: May 24, 2020

Heparin failure and COVID-19: Should we explore other anticoagulants? An observational report regarding in-vitro recovery of anticoagulant action in COVID-19 patients in intensive care.

Heparin failure and COVID-19: Should we explore other anticoagulants? An observational report regarding in-vitro recovery of anticoagulant action in COVID-19 patients in intensive care.

Journal: Thrombosis research

Published: May 19, 2020

Molecular Simulation of αvβ6 Integrin Inhibitors.

Molecular Simulation of αvβ6 Integrin Inhibitors.

Journal: Journal of chemical information and modeling

Published: May 19, 2020

Showing 1-12 of 51

Last Updated: 09/26/2026